Kumar A - Search Results

1

Novel 1,2,4-triazoles as selective carbonic anhydrase inhibitors showing ancillary anticathepsin B activity.

Kumar A, Arya P, Giovannuzzi S, Mohan B, Raghav N, Supuran CT, Sharma PK. Kumar A, et al. Future Med Chem. 2024 Apr 4. doi: 10.4155/fmc-2023-0321. Online ahead of print. Future Med Chem. 2024. PMID: 38573017

2

A decade of tail-approach based design of selective as well as potent tumor associated carbonic anhydrase inhibitors.

Kumar A, Siwach K, Supuran CT, Sharma PK. Kumar A, et al. Bioorg Chem. 2022 Sep;126:105920. doi: 10.1016/j.bioorg.2022.105920. Epub 2022 Jun 1. Bioorg Chem. 2022. PMID: 35671645 Review.

3

Novel benzenesulfonamide-bearing pyrazoles and 1,2,4-thiadiazoles as selective carbonic anhydrase inhibitors.

Kumar R, Kumar A, Ram S, Angeli A, Bonardi A, Nocentini A, Gratteri P, Supuran CT, Sharma PK. Kumar R, et al. Among authors: kumar a. Arch Pharm (Weinheim). 2022 Jan;355(1):e2100241. doi: 10.1002/ardp.202100241. Epub 2021 Oct 1. Arch Pharm (Weinheim). 2022. PMID: 34596922

4

Tail-approach based design and synthesis of Arylthiazolylhydrazono-1,2,3-triazoles incorporating sulfanilamide and metanilamide as human carbonic anhydrase I, II, IV and IX inhibitors.

Kumar A, Siwach K, Rom T, Kumar R, Angeli A, Kumar Paul A, Supuran CT, Sharma PK. Kumar A, et al. Among authors: kumar paul a, kumar r. Bioorg Chem. 2022 Jun;123:105764. doi: 10.1016/j.bioorg.2022.105764. Epub 2022 Mar 26. Bioorg Chem. 2022. PMID: 35366582

5

Selective inhibition of carbonic anhydrase IX by sulphonylated 1,2,3-triazole incorporated benzenesulphonamides capable of inducing apoptosis.

Siwach K, Kumar A, Panchal H, Kumar R, Bhardwaj JK, Angeli A, Supuran CT, Sharma PK. Siwach K, et al. Among authors: kumar r, kumar a. J Enzyme Inhib Med Chem. 2022 Dec;37(1):1454-1463. doi: 10.1080/14756366.2022.2077333. J Enzyme Inhib Med Chem. 2022. PMID: 35616287 Free PMC article.

6

Potent inhibitors of tumor associated carbonic anhydrases endowed with cathepsin B inhibition.

Kumar A, Arya P, Sharma V, Giovannuzzi S, Raghav N, Supuran CT, Sharma PK. Kumar A, et al. Arch Pharm (Weinheim). 2023 Nov;356(11):e2300349. doi: 10.1002/ardp.202300349. Epub 2023 Sep 13. Arch Pharm (Weinheim). 2023. PMID: 37704930

7

Synthesis, Structure-Activity Relationships, and In Vivo Evaluation of Novel Tetrahydropyran-Based Thiodisaccharide Mimics as Galectin-3 Inhibitors.

Xu L, Hartz RA, Beno BR, Ghosh K, Shukla JK, Kumar A, Patel D, Kalidindi N, Lemos N, Gautam SS, Kumar A, Ellsworth BA, Shah D, Sale H, Cheng D, Regueiro-Ren A. Xu L, et al. Among authors: kumar a. J Med Chem. 2021 May 27;64(10):6634-6655. doi: 10.1021/acs.jmedchem.0c02001. Epub 2021 May 14. J Med Chem. 2021. PMID: 33988358

8

Synthesis, Computational and Pharmacological Evaluation of 7-(2-(2- (3- (Substituted Phenyl) Acryloyl) Phenoxy) Ethoxy)-4-Methyl-2H-Chromen- 2-Ones as CNS Agents.

Kumar S, Kumar A. Kumar S, et al. Among authors: kumar a. Cent Nerv Syst Agents Med Chem. 2023;23(1):57-64. doi: 10.2174/1871524923666230130134501. Cent Nerv Syst Agents Med Chem. 2023. PMID: 36717998

9

Microtubule stabilising peptides: new paradigm towards management of neuronal disorders.

Bhargava S, Kulkarni R, Dewangan B, Kulkarni N, Jiaswar C, Kumar K, Kumar A, Bodhe PR, Kumar H, Sahu B. Bhargava S, et al. Among authors: kumar k, kumar h, kumar a. RSC Med Chem. 2023 Aug 14;14(11):2192-2205. doi: 10.1039/d3md00012e. eCollection 2023 Nov 15. RSC Med Chem. 2023. PMID: 37974959 Review.

10

Discovery of BMS-986144, a Third-Generation, Pan-Genotype NS3/4A Protease Inhibitor for the Treatment of Hepatitis C Virus Infection.

Sun LQ, Mull E, D'Andrea S, Zheng B, Hiebert S, Gillis E, Bowsher M, Kandhasamy S, Baratam VR, Puttaswamy S, Pulicharla N, Vishwakrishnan S, Reddy S, Trivedi R, Sinha S, Sivaprasad S, Rao A, Desai S, Ghosh K, Anumula R, Kumar A, Rajamani R, Wang YK, Fang H, Mathur A, Rampulla R, Zvyaga TA, Mosure K, Jenkins S, Falk P, Tagore DM, Chen C, Rendunchintala K, Loy J, Meanwell NA, McPhee F, Scola PM. Sun LQ, et al. Among authors: kumar a. J Med Chem. 2020 Dec 10;63(23):14740-14760. doi: 10.1021/acs.jmedchem.0c01296. Epub 2020 Nov 23. J Med Chem. 2020. PMID: 33226226

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