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Novel-Type GABAB PAMs: Structure-Activity Relationship in Light of the Protein Structure.
ACS Med Chem Lett. 2024 Mar 1;15(3):396-405. doi: 10.1021/acsmedchemlett.3c00560. eCollection 2024 Mar 14.
ACS Med Chem Lett. 2024.
PMID: 38505850
Multiparameter Optimization of Naphthyridine Derivatives as Selective α5-GABAA Receptor Negative Allosteric Modulators.
Szabó G, Éliás O, Erdélyi P, Potor A, Túrós GI, Károlyi BI, Varró G, Vaskó ÁG, Bata I, Kapus GL, Dohányos Z, Bobok AÁ, Fodor L, Thán M, Vastag M, Komlódi Z, Soukupné Kedves RÉ, Makó É, Süveges B, Greiner I.
Szabó G, et al. Among authors: bobok aa.
J Med Chem. 2022 Jun 9;65(11):7876-7895. doi: 10.1021/acs.jmedchem.2c00414. Epub 2022 May 18.
J Med Chem. 2022.
PMID: 35584373
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6-Aryl-quinazolines as novel GABAB receptor positive allosteric modulators.
Huszár J, Petró JL, Hadady Z, Bobok AÁ, Sághy K, Halász AS, Hornyánszky G, Román V, Greiner I, Éles J.
Huszár J, et al. Among authors: bobok aa.
Bioorg Med Chem Lett. 2022 Jul 1;67:128714. doi: 10.1016/j.bmcl.2022.128714. Epub 2022 Apr 1.
Bioorg Med Chem Lett. 2022.
PMID: 35367591
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