Discovery of Novel 5,6-Dihydro-4H-pyrido[2,3,4-de]quinazoline Irreversible Inhibitors Targeting Both Wild-Type and A775_G776insYVMA Mutated HER2 Kinases.
Yang L, Li Y, Du Y, Guo Y, Guo Z, Liu B, Liu J, Liu Y, Niu H, Sun Y, Yan H, Yang Y, Yu S, Zhang Y, Zhang Y, Zheng K, Zheng N, Zhang X, Zhang Q, Hu L.
Yang L, et al. Among authors: liu j, liu y, liu b.
J Med Chem. 2024 Apr 11;67(7):5662-5682. doi: 10.1021/acs.jmedchem.3c02302. Epub 2024 Mar 22.
J Med Chem. 2024.
PMID: 38518121