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Design, synthesis, ADME and biological evaluation of benzylpiperidine and benzylpiperazine derivatives as novel reversible monoacylglycerol lipase (MAGL) inhibitors.
Di Stefano M, Masoni S, Bononi G, Poli G, Galati S, Gado F, Manzi S, Vagaggini C, Brai A, Caligiuri I, Asif K, Rizzolio F, Macchia M, Chicca A, Sodi A, Di Bussolo V, Minutolo F, Meier P, Gertsch J, Granchi C, Dreassi E, Tuccinardi T. Di Stefano M, et al. Among authors: bononi g. Eur J Med Chem. 2024 Jan 5;263:115916. doi: 10.1016/j.ejmech.2023.115916. Epub 2023 Nov 2. Eur J Med Chem. 2024. PMID: 37976705 Free article.
Machine Learning-Based Virtual Screening for the Identification of Cdk5 Inhibitors.
Di Stefano M, Galati S, Ortore G, Caligiuri I, Rizzolio F, Ceni C, Bertini S, Bononi G, Granchi C, Macchia M, Poli G, Tuccinardi T. Di Stefano M, et al. Among authors: bononi g. Int J Mol Sci. 2022 Sep 13;23(18):10653. doi: 10.3390/ijms231810653. Int J Mol Sci. 2022. PMID: 36142566 Free PMC article.
Reversible Monoacylglycerol Lipase Inhibitors: Discovery of a New Class of Benzylpiperidine Derivatives.
Bononi G, Di Stefano M, Poli G, Ortore G, Meier P, Masetto F, Caligiuri I, Rizzolio F, Macchia M, Chicca A, Avan A, Giovannetti E, Vagaggini C, Brai A, Dreassi E, Valoti M, Minutolo F, Granchi C, Gertsch J, Tuccinardi T. Bononi G, et al. J Med Chem. 2022 May 26;65(10):7118-7140. doi: 10.1021/acs.jmedchem.1c01806. Epub 2022 May 6. J Med Chem. 2022. PMID: 35522977 Free PMC article.
18 results