Fischer S - Search Results

1

Preclinical evaluation of an ¹⁸F-labeled N^ε-acryloyllysine piperazide for covalent targeting of transglutaminase 2.

Wodtke R, Laube M, Hauser S, Meister S, Ludwig FA, Fischer S, Kopka K, Pietzsch J, Löser R. Wodtke R, et al. Among authors: fischer s. EJNMMI Radiopharm Chem. 2024 Jan 2;9(1):1. doi: 10.1186/s41181-023-00231-1. EJNMMI Radiopharm Chem. 2024. PMID: 38165538 Free PMC article.

2

N^ε-Acryloyllysine Piperazides as Irreversible Inhibitors of Transglutaminase 2: Synthesis, Structure-Activity Relationships, and Pharmacokinetic Profiling.

Wodtke R, Hauser C, Ruiz-Gómez G, Jäckel E, Bauer D, Lohse M, Wong A, Pufe J, Ludwig FA, Fischer S, Hauser S, Greif D, Pisabarro MT, Pietzsch J, Pietsch M, Löser R. Wodtke R, et al. Among authors: fischer s. J Med Chem. 2018 May 24;61(10):4528-4560. doi: 10.1021/acs.jmedchem.8b00286. Epub 2018 May 10. J Med Chem. 2018. PMID: 29664627

3

Development of ¹⁸F-Labeled Radiotracers for PET Imaging of the Adenosine A_2A Receptor: Synthesis, Radiolabeling and Preliminary Biological Evaluation.

Lai TH, Schröder S, Toussaint M, Dukić-Stefanović S, Kranz M, Ludwig FA, Fischer S, Steinbach J, Deuther-Conrad W, Brust P, Moldovan RP. Lai TH, et al. Among authors: fischer s. Int J Mol Sci. 2021 Feb 25;22(5):2285. doi: 10.3390/ijms22052285. Int J Mol Sci. 2021. PMID: 33669003 Free PMC article.

4

Design, Radiosynthesis and Preliminary Biological Evaluation in Mice of a Brain-Penetrant ¹⁸F-Labelled σ₂ Receptor Ligand.

Moldovan RP, Gündel D, Teodoro R, Ludwig FA, Fischer S, Toussaint M, Schepmann D, Wünsch B, Brust P, Deuther-Conrad W. Moldovan RP, et al. Among authors: fischer s. Int J Mol Sci. 2021 May 21;22(11):5447. doi: 10.3390/ijms22115447. Int J Mol Sci. 2021. PMID: 34064122 Free PMC article.

5

Radiosynthesis of (S)-[¹⁸F]T1: The first PET radioligand for molecular imaging of α3β4 nicotinic acetylcholine receptors.

Sarasamkan J, Fischer S, Deuther-Conrad W, Ludwig FA, Scheunemann M, Arunrungvichian K, Vajragupta O, Brust P. Sarasamkan J, et al. Among authors: fischer s. Appl Radiat Isot. 2017 Jun;124:106-113. doi: 10.1016/j.apradiso.2017.03.015. Epub 2017 Mar 18. Appl Radiat Isot. 2017. PMID: 28365525

6

Exploring the Metabolism of (+)-[¹⁸F]Flubatine in Vitro and in Vivo: LC-MS/MS Aided Identification of Radiometabolites in a Clinical PET Study.

Ludwig FA, Fischer S, Smits R, Deuther-Conrad W, Hoepping A, Tiepolt S, Patt M, Sabri O, Brust P. Ludwig FA, et al. Among authors: fischer s. Molecules. 2018 Feb 20;23(2):464. doi: 10.3390/molecules23020464. Molecules. 2018. PMID: 29461507 Free PMC article.

7

Asymmetric Synthesis of Spirocyclic 2-Benzopyrans for Positron Emission Tomography of σ1 Receptors in the Brain.

Holl K, Schepmann D, Fischer S, Ludwig FA, Hiller A, Donat CK, Deuther-Conrad W, Brust P, Wünsch B. Holl K, et al. Among authors: fischer s. Pharmaceuticals (Basel). 2014 Jan 22;7(1):78-112. doi: 10.3390/ph7010078. Pharmaceuticals (Basel). 2014. PMID: 24451404 Free PMC article.

8

Development of a Novel Nonpeptidic (18)F-Labeled Radiotracer for in Vivo Imaging of Oxytocin Receptors with Positron Emission Tomography.

Wenzel B, Mollitor J, Deuther-Conrad W, Dukic-Stefanovic S, Kranz M, Vraka C, Teodoro R, Günther R, Donat CK, Ludwig FA, Fischer S, Smits R, Wadsak W, Mitterhauser M, Steinbach J, Hoepping A, Brust P. Wenzel B, et al. Among authors: fischer s. J Med Chem. 2016 Mar 10;59(5):1800-17. doi: 10.1021/acs.jmedchem.5b01080. Epub 2016 Feb 3. J Med Chem. 2016. PMID: 26796795

9

LC-MS Supported Studies on the in Vitro Metabolism of both Enantiomers of Flubatine and the in Vivo Metabolism of (+)-[(18)F]Flubatine-A Positron Emission Tomography Radioligand for Imaging α4β2 Nicotinic Acetylcholine Receptors.

Ludwig FA, Smits R, Fischer S, Donat CK, Hoepping A, Brust P, Steinbach J. Ludwig FA, et al. Among authors: fischer s. Molecules. 2016 Sep 8;21(9):1200. doi: 10.3390/molecules21091200. Molecules. 2016. PMID: 27617996 Free PMC article.

10

Bridging from Brain to Tumor Imaging: (S)-(-)- and (R)-(+)-[¹⁸F]Fluspidine for Investigation of Sigma-1 Receptors in Tumor-Bearing Mice.

Kranz M, Bergmann R, Kniess T, Belter B, Neuber C, Cai Z, Deng G, Fischer S, Zhou J, Huang Y, Brust P, Deuther-Conrad W, Pietzsch J. Kranz M, et al. Among authors: fischer s. Molecules. 2018 Mar 20;23(3):702. doi: 10.3390/molecules23030702. Molecules. 2018. PMID: 29558382 Free PMC article.

Save citations to file

Email citations

Send citations to clipboard

Add to Collections

Add to My Bibliography

Create a file for external citation management software

Your saved search

Your RSS Feed

My NCBI Filters

Text availability

Article attribute

Article type

Publication date

3,678 results

Search Page