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New azaaurone derivatives as potential multitarget agents in HIV-TB coinfection.
Arch Pharm (Weinheim). 2024 Feb;357(2):e2300560. doi: 10.1002/ardp.202300560. Epub 2023 Nov 30.
Arch Pharm (Weinheim). 2024.
PMID: 38032154
Drug discovery in tuberculosis. New drug targets and antimycobacterial agents.
Campaniço A, Moreira R, Lopes F.
Campaniço A, et al.
Eur J Med Chem. 2018 Apr 25;150:525-545. doi: 10.1016/j.ejmech.2018.03.020. Epub 2018 Mar 9.
Eur J Med Chem. 2018.
PMID: 29549838
Review.
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Azaaurones as Potent Antimycobacterial Agents Active against MDR- and XDR-TB.
Campaniço A, Carrasco MP, Njoroge M, Seldon R, Chibale K, Perdigão J, Portugal I, Warner DF, Moreira R, Lopes F.
Campaniço A, et al.
ChemMedChem. 2019 Aug 20;14(16):1537-1546. doi: 10.1002/cmdc.201900289. Epub 2019 Jul 25.
ChemMedChem. 2019.
PMID: 31294529
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Addressing Latent Tuberculosis: New Advances in Mimicking the Disease, Discovering Key Targets, and Designing Hit Compounds.
Campaniço A, Harjivan SG, Warner DF, Moreira R, Lopes F.
Campaniço A, et al.
Int J Mol Sci. 2020 Nov 23;21(22):8854. doi: 10.3390/ijms21228854.
Int J Mol Sci. 2020.
PMID: 33238468
Free PMC article.
Review.
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Structural Optimization of Antimycobacterial Azaaurones Towards Improved Solubility and Metabolic Stability.
Campaniço A, Harjivan SG, Freitas E, Serafini M, Gaspar MM, Capela R, Gomes P, Jordaan A, Madureira AM, André V, Silva AB, Duarte MT, Portugal I, Perdigão J, Moreira R, Warner DF, Lopes F.
Campaniço A, et al.
ChemMedChem. 2023 Dec 14;18(24):e202300410. doi: 10.1002/cmdc.202300410. Epub 2023 Nov 6.
ChemMedChem. 2023.
PMID: 37845182
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