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Novel Kinetic Resolution of Thiazolo-Benzimidazolines Using MAO Enzymes.
ACS Omega. 2023 Nov 1;8(45):42114-42125. doi: 10.1021/acsomega.3c03223. eCollection 2023 Nov 14.
ACS Omega. 2023.
PMID: 38024698
Free PMC article.
Structure-Based Bioisosterism Design, Synthesis, Biological Evaluation and In Silico Studies of Benzamide Analogs as Potential Anthelmintics.
Vairoletti F, Paulino M, Mahler G, Salinas G, Saiz C.
Vairoletti F, et al.
Molecules. 2022 Apr 20;27(9):2659. doi: 10.3390/molecules27092659.
Molecules. 2022.
PMID: 35566007
Free PMC article.
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Increased sensitivity of an infrared motility assay for nematicide discovery.
Vairoletti F, Baron A, Saiz C, Mahler G, Salinas G.
Vairoletti F, et al.
MicroPubl Biol. 2021 Nov 30;2021:10.17912/micropub.biology.000500. doi: 10.17912/micropub.biology.000500. eCollection 2021.
MicroPubl Biol. 2021.
PMID: 34870110
Free PMC article.
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A multiscale approach to predict the binding mode of metallo beta-lactamase inhibitors.
Gervasoni S, Spencer J, Hinchliffe P, Pedretti A, Vairoletti F, Mahler G, Mulholland AJ.
Gervasoni S, et al. Among authors: vairoletti f.
Proteins. 2022 Feb;90(2):372-384. doi: 10.1002/prot.26227. Epub 2021 Sep 20.
Proteins. 2022.
PMID: 34455628
Free PMC article.
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Synthesis of bicyclic 1,4-thiazepines as novel anti-Trypanosoma brucei brucei agents.
Vairoletti F, Medeiros A, Fontán P, Meléndrez J, Tabárez C, Salinas G, Franco J, Comini MA, Saldaña J, Jancik V, Mahler G, Saiz C.
Vairoletti F, et al.
Medchemcomm. 2019 Jun 11;10(8):1481-1487. doi: 10.1039/c9md00064j. eCollection 2019 Aug 1.
Medchemcomm. 2019.
PMID: 31673311
Free PMC article.
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