Search Page
Save citations to file
Email citations
Send citations to clipboard
Add to Collections
Add to My Bibliography
Create a file for external citation management software
Your saved search
Your RSS Feed
Search Results
8 results
Filters applied: . Clear all
Results are displayed in a computed author sort order.
The Results By Year timeline is not available.
Page 1
Covalent Stapling of the Cereblon Sensor Loop Histidine Using Sulfur-Heterocycle Exchange.
ACS Med Chem Lett. 2023 Oct 24;14(11):1576-1581. doi: 10.1021/acsmedchemlett.3c00371. eCollection 2023 Nov 9.
ACS Med Chem Lett. 2023.
PMID: 37974938
HiBiT-SpyTag: A Minimal Tag for Covalent Protein Capture and Degrader Development.
Tsang T, Huerta F, Liu Y, Che J, Metivier RJ, Ferrao S, Donovan KA, Jones LH, Zerfas BL, Nowak RP.
Tsang T, et al. Among authors: metivier rj.
ACS Chem Biol. 2023 Apr 21;18(4):933-941. doi: 10.1021/acschembio.3c00084. Epub 2023 Apr 5.
ACS Chem Biol. 2023.
PMID: 37018062
Item in Clipboard
Catalytic Degraders Effectively Address Kinase Site Mutations in EML4-ALK Oncogenic Fusions.
Gao Y, Jiang B, Kim H, Berberich MJ, Che J, Donovan KA, Hatcher JM, Huerta F, Kwiatkowski NP, Liu Y, Liuni PP, Metivier RJ, Murali VK, Nowak RP, Zhang T, Fischer ES, Gray NS, Jones LH.
Gao Y, et al. Among authors: metivier rj.
J Med Chem. 2023 Apr 27;66(8):5524-5535. doi: 10.1021/acs.jmedchem.2c01864. Epub 2023 Apr 10.
J Med Chem. 2023.
PMID: 37036171
Item in Clipboard
Development of a covalent cereblon-based PROTAC employing a fluorosulfate warhead.
Nowak RP, Ragosta L, Huerta F, Liu H, Ficarro SB, Cruite JT, Metivier RJ, Donovan KA, Marto JA, Fischer ES, Zerfas BL, Jones LH.
Nowak RP, et al. Among authors: metivier rj.
RSC Chem Biol. 2023 Aug 31;4(11):906-912. doi: 10.1039/d3cb00103b. eCollection 2023 Nov 1.
RSC Chem Biol. 2023.
PMID: 37920397
Free PMC article.
Item in Clipboard
Development of sulfonyl fluoride chemical probes to advance the discovery of cereblon modulators.
Liu Y, Nowak RP, Che J, Donovan KA, Huerta F, Liu H, Metivier RJ, Fischer ES, Jones LH.
Liu Y, et al. Among authors: metivier rj.
RSC Med Chem. 2024 Jan 9;15(2):607-611. doi: 10.1039/d3md00652b. eCollection 2024 Feb 21.
RSC Med Chem. 2024.
PMID: 38389883
Item in Clipboard
Discovery of CRBN-dependent WEE1 Molecular Glue Degraders from a Multicomponent Combinatorial Library.
Razumkov H, Jiang Z, Baek K, You I, Geng Q, Donovan KA, Tang MT, Metivier RJ, Mageed N, Seo P, Li Z, Byun WS, Hinshaw SM, Sarott RC, Fischer ES, Gray NS.
Razumkov H, et al. Among authors: metivier rj.
bioRxiv [Preprint]. 2024 May 5:2024.05.04.592550. doi: 10.1101/2024.05.04.592550.
bioRxiv. 2024.
PMID: 38746375
Free PMC article.
Preprint.
Item in Clipboard
Characterization of Serine Hydrolases Across Clinical Isolates of Commensal Skin Bacteria Staphylococcus epidermidis Using Activity-Based Protein Profiling.
Keller LJ, Lentz CS, Chen YE, Metivier RJ, Weerapana E, Fischbach MA, Bogyo M.
Keller LJ, et al. Among authors: metivier rj.
ACS Infect Dis. 2020 May 8;6(5):930-938. doi: 10.1021/acsinfecdis.0c00095. Epub 2020 Apr 27.
ACS Infect Dis. 2020.
PMID: 32298574
Item in Clipboard
Cereblon covalent modulation through structure-based design of histidine targeting chemical probes.
Cruite JT, Dann GP, Che J, Donovan KA, Ferrao S, Ficarro SB, Fischer ES, Gray NS, Huerta F, Kong NR, Liu H, Marto JA, Metivier RJ, Nowak RP, Zerfas BL, Jones LH.
Cruite JT, et al. Among authors: metivier rj.
RSC Chem Biol. 2022 Jul 8;3(9):1105-1110. doi: 10.1039/d2cb00078d. eCollection 2022 Aug 31.
RSC Chem Biol. 2022.
PMID: 36128501
Free PMC article.
Item in Clipboard
Cite
Cite