Alt J - Search Results

1

Discovery of tert-Butyl Ester Based 6-Diazo-5-oxo-l-norleucine Prodrugs for Enhanced Metabolic Stability and Tumor Delivery.

Novotná K, Tenora L, Prchalová E, Paule J, Alt J, Veeravalli V, Lam J, Wu Y, Šnajdr I, Gori S, Mettu VS, Tsukamoto T, Majer P, Slusher BS, Rais R. Novotná K, et al. Among authors: alt j. J Med Chem. 2023 Nov 23;66(22):15493-15510. doi: 10.1021/acs.jmedchem.3c01681. Epub 2023 Nov 10. J Med Chem. 2023. PMID: 37949450 Free PMC article.

2

Inhibition of xc⁻ transporter-mediated cystine uptake by sulfasalazine analogs.

Shukla K, Thomas AG, Ferraris DV, Hin N, Sattler R, Alt J, Rojas C, Slusher BS, Tsukamoto T. Shukla K, et al. Among authors: alt j. Bioorg Med Chem Lett. 2011 Oct 15;21(20):6184-7. doi: 10.1016/j.bmcl.2011.07.081. Epub 2011 Aug 12. Bioorg Med Chem Lett. 2011. PMID: 21889337

3

Development of a high-throughput method for the determination of pharmacological levels of plasma D-serine.

Alt J, Rojas C, Wozniak K, Wu Y, Ferraris D, Tsukamoto T, Slusher B. Alt J, et al. Anal Biochem. 2011 Dec 15;419(2):106-9. doi: 10.1016/j.ab.2011.08.018. Epub 2011 Aug 16. Anal Biochem. 2011. PMID: 21889486 Free PMC article.

4

Reversible disulfide formation of the glutamate carboxypeptidase II inhibitor E2072 results in prolonged systemic exposures in vivo.

Rais R, Hoover R, Wozniak K, Rudek MA, Tsukamoto T, Alt J, Rojas C, Slusher BS. Rais R, et al. Among authors: alt j. Drug Metab Dispos. 2012 Dec;40(12):2315-23. doi: 10.1124/dmd.112.046821. Epub 2012 Sep 4. Drug Metab Dispos. 2012. PMID: 22949627 Free PMC article.

5

Design, synthesis, and pharmacological evaluation of bis-2-(5-phenylacetamido-1,2,4-thiadiazol-2-yl)ethyl sulfide 3 (BPTES) analogs as glutaminase inhibitors.

Shukla K, Ferraris DV, Thomas AG, Stathis M, Duvall B, Delahanty G, Alt J, Rais R, Rojas C, Gao P, Xiang Y, Dang CV, Slusher BS, Tsukamoto T. Shukla K, et al. Among authors: alt j. J Med Chem. 2012 Dec 13;55(23):10551-63. doi: 10.1021/jm301191p. Epub 2012 Nov 30. J Med Chem. 2012. PMID: 23151085 Free PMC article.

6

Synthesis and SAR of 1-hydroxy-1H-benzo[d]imidazol-2(3H)-ones as Inhibitors of D-Amino Acid Oxidase.

Berry JF, Ferraris DV, Duvall B, Hin N, Rais R, Alt J, Thomas AG, Rojas C, Hashimoto K, Slusher BS, Tsukamoto T. Berry JF, et al. Among authors: alt j. ACS Med Chem Lett. 2012 Oct 11;3(10):839-843. doi: 10.1021/ml300212a. Epub 2012 Sep 16. ACS Med Chem Lett. 2012. PMID: 23243487 Free PMC article.

7

Synthesis of kojic acid derivatives as secondary binding site probes of D-amino acid oxidase.

Raje M, Hin N, Duvall B, Ferraris DV, Berry JF, Thomas AG, Alt J, Rojas C, Slusher BS, Tsukamoto T. Raje M, et al. Among authors: alt j. Bioorg Med Chem Lett. 2013 Jul 1;23(13):3910-3. doi: 10.1016/j.bmcl.2013.04.062. Epub 2013 May 1. Bioorg Med Chem Lett. 2013. PMID: 23683589 Free PMC article.

8

δ-Thiolactones as prodrugs of thiol-based glutamate carboxypeptidase II (GCPII) inhibitors.

Ferraris DV, Majer P, Ni C, Slusher CE, Rais R, Wu Y, Wozniak KM, Alt J, Rojas C, Slusher BS, Tsukamoto T. Ferraris DV, et al. Among authors: alt j. J Med Chem. 2014 Jan 9;57(1):243-7. doi: 10.1021/jm401703a. Epub 2013 Dec 27. J Med Chem. 2014. PMID: 24354364 Free PMC article.

9

Design, synthesis, and pharmacological evaluation of fluorinated tetrahydrouridine derivatives as inhibitors of cytidine deaminase.

Ferraris D, Duvall B, Delahanty G, Mistry B, Alt J, Rojas C, Rowbottom C, Sanders K, Schuck E, Huang KC, Redkar S, Slusher BB, Tsukamoto T. Ferraris D, et al. Among authors: alt j. J Med Chem. 2014 Mar 27;57(6):2582-8. doi: 10.1021/jm401856k. Epub 2014 Feb 24. J Med Chem. 2014. PMID: 24520856

10

Peptidomimetics of Arg-Phe-NH2 as small molecule agonists of Mas-related gene C (MrgC) receptors.

Hin N, Alt J, Zimmermann SC, Delahanty G, Ferraris DV, Rojas C, Li F, Liu Q, Dong X, Slusher BS, Tsukamoto T. Hin N, et al. Among authors: alt j. Bioorg Med Chem. 2014 Nov 1;22(21):5831-7. doi: 10.1016/j.bmc.2014.09.025. Epub 2014 Sep 19. Bioorg Med Chem. 2014. PMID: 25288495 Free PMC article.

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