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Structure-Based Drug Discovery with Deep Learning.
Özçelik R, van Tilborg D, Jiménez-Luna J, Grisoni F. Özçelik R, et al. Among authors: grisoni f. Chembiochem. 2023 Jul 3;24(13):e202200776. doi: 10.1002/cbic.202200776. Epub 2023 Jun 13. Chembiochem. 2023. PMID: 37014633 Review.
Deep learning for low-data drug discovery: Hurdles and opportunities.
van Tilborg D, Brinkmann H, Criscuolo E, Rossen L, Özçelik R, Grisoni F. van Tilborg D, et al. Among authors: grisoni f. Curr Opin Struct Biol. 2024 Jun;86:102818. doi: 10.1016/j.sbi.2024.102818. Epub 2024 Apr 25. Curr Opin Struct Biol. 2024. PMID: 38669740 Free article. Review.
Is Antipsychotic Drug Use During Pregnancy Associated with Increased Malformation Rates and Worsening of Maternal and Infant Outcomes? A Systematic Review.
Sani G, Callovini T, Ferrara OM, Segatori D, Margoni S, Simonetti A, Lisci FM, Marano G, Fischetti A, Kotzalidis GD, Di Segni F, Fiaschè F, Janiri D, Moccia L, Manfredi G, Alcibiade A, Brisi C, Grisoni F, Stella G, Bernardi E, Brugnami A, Ciliberto M, Spera MC, Caso R, Rossi S, Boggio G, Mastroeni G, Abate F, Conte E, Quintano A, De Chiara L, Monti L, Camardese G, Rinaldi L, Koukopoulos AE, Chieffo DPR, Angeletti G, Mazza M. Sani G, et al. Among authors: grisoni f. Curr Neuropharmacol. 2024 May 17. doi: 10.2174/1570159X22666240516151449. Online ahead of print. Curr Neuropharmacol. 2024. PMID: 38766824
Baricitinib and tofacitinib off-target profile, with a focus on Alzheimer's disease.
Faquetti ML, Slappendel L, Bigonne H, Grisoni F, Schneider P, Aichinger G, Schneider G, Sturla SJ, Burden AM. Faquetti ML, et al. Among authors: grisoni f. Alzheimers Dement (N Y). 2024 Jan 26;10(1):e12445. doi: 10.1002/trc2.12445. eCollection 2024 Jan-Mar. Alzheimers Dement (N Y). 2024. PMID: 38528988 Free PMC article.
Artificial intelligence for natural product drug discovery.
Mullowney MW, Duncan KR, Elsayed SS, Garg N, van der Hooft JJJ, Martin NI, Meijer D, Terlouw BR, Biermann F, Blin K, Durairaj J, Gorostiola González M, Helfrich EJN, Huber F, Leopold-Messer S, Rajan K, de Rond T, van Santen JA, Sorokina M, Balunas MJ, Beniddir MA, van Bergeijk DA, Carroll LM, Clark CM, Clevert DA, Dejong CA, Du C, Ferrinho S, Grisoni F, Hofstetter A, Jespers W, Kalinina OV, Kautsar SA, Kim H, Leao TF, Masschelein J, Rees ER, Reher R, Reker D, Schwaller P, Segler M, Skinnider MA, Walker AS, Willighagen EL, Zdrazil B, Ziemert N, Goss RJM, Guyomard P, Volkamer A, Gerwick WH, Kim HU, Müller R, van Wezel GP, van Westen GJP, Hirsch AKH, Linington RG, Robinson SL, Medema MH. Mullowney MW, et al. Among authors: grisoni f. Nat Rev Drug Discov. 2023 Nov;22(11):895-916. doi: 10.1038/s41573-023-00774-7. Epub 2023 Sep 11. Nat Rev Drug Discov. 2023. PMID: 37697042 Review.
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