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Fragment expansion with NUDELs - poised DNA-encoded libraries.
Chem Sci. 2023 Jul 12;14(31):8288-8294. doi: 10.1039/d3sc01171b. eCollection 2023 Aug 9.
Chem Sci. 2023.
PMID: 37564419
Free PMC article.
On the design of lead-like DNA-encoded chemical libraries.
Castan IFSF, Graham JS, Salvini CLA, Stanway-Gordon HA, Waring MJ.
Castan IFSF, et al. Among authors: salvini cla.
Bioorg Med Chem. 2021 Aug 1;43:116273. doi: 10.1016/j.bmc.2021.116273. Epub 2021 Jun 10.
Bioorg Med Chem. 2021.
PMID: 34147943
Review.
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Highly efficient on-DNA amide couplings promoted by micelle forming surfactants for the synthesis of DNA encoded libraries.
Hunter JH, Anderson MJ, Castan IFSF, Graham JS, Salvini CLA, Stanway-Gordon HA, Crawford JJ, Madin A, Pairaudeau G, Waring MJ.
Hunter JH, et al. Among authors: salvini cla.
Chem Sci. 2021 Jun 22;12(27):9475-9484. doi: 10.1039/d1sc03007h. eCollection 2021 Jul 14.
Chem Sci. 2021.
PMID: 34349922
Free PMC article.
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Micelle-Promoted Reductive Amination of DNA-Conjugated Amines for DNA-Encoded Library Synthesis.
Anderson MJ, Carton TP, Salvini CLA, Crawford JJ, Pairaudeau G, Waring MJ.
Anderson MJ, et al. Among authors: salvini cla.
Chemistry. 2024 Apr 11;30(21):e202400239. doi: 10.1002/chem.202400239. Epub 2024 Feb 21.
Chemistry. 2024.
PMID: 38251309
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