Almqvist F - Search Results

1

Design, Synthesis, and Evaluation of Novel Δ²-Thiazolino 2-Pyridone Derivatives That Potentiate Isoniazid Activity in an Isoniazid-Resistant Mycobacterium tuberculosis Mutant.

Sarkar S, Mayer Bridwell AE, Good JAD, Wang ER, McKee SR, Valenta J, Harrison GA, Flentie KN, Henry FL, Wixe T, Demirel P, Vagolu SK, Chatagnon J, Machelart A, Brodin P, Tønjum T, Stallings CL, Almqvist F. Sarkar S, et al. Among authors: almqvist f. J Med Chem. 2023 Aug 24;66(16):11056-11077. doi: 10.1021/acs.jmedchem.3c00358. Epub 2023 Jul 24. J Med Chem. 2023. PMID: 37485869 Free PMC article.

2

Multivariate design, synthesis, and biological evaluation of peptide inhibitors of FimC/FimH protein-protein interactions in uropathogenic Escherichia coli.

Larsson A, Johansson SM, Pinkner JS, Hultgren SJ, Almqvist F, Kihlberg J, Linusson A. Larsson A, et al. Among authors: almqvist f. J Med Chem. 2005 Feb 24;48(4):935-45. doi: 10.1021/jm040818l. J Med Chem. 2005. PMID: 15715464

3

Design, synthesis and evaluation of peptidomimetics based on substituted bicyclic 2-pyridones-targeting virulence of uropathogenic E. coli.

Berg V, Sellstedt M, Hedenström M, Pinkner JS, Hultgren SJ, Almqvist F. Berg V, et al. Among authors: almqvist f. Bioorg Med Chem. 2006 Nov 15;14(22):7563-81. doi: 10.1016/j.bmc.2006.07.017. Epub 2006 Aug 14. Bioorg Med Chem. 2006. PMID: 16904898

4

Design and synthesis of C-2 substituted thiazolo and dihydrothiazolo ring-fused 2-pyridones: pilicides with increased antivirulence activity.

Chorell E, Pinkner JS, Phan G, Edvinsson S, Buelens F, Remaut H, Waksman G, Hultgren SJ, Almqvist F. Chorell E, et al. Among authors: almqvist f. J Med Chem. 2010 Aug 12;53(15):5690-5. doi: 10.1021/jm100470t. J Med Chem. 2010. PMID: 20586493 Free PMC article.

5

Synthesis and application of a bromomethyl substituted scaffold to be used for efficient optimization of anti-virulence activity.

Chorell E, Bengtsson C, Sainte-Luce Banchelin T, Das P, Uvell H, Sinha AK, Pinkner JS, Hultgren SJ, Almqvist F. Chorell E, et al. Among authors: almqvist f. Eur J Med Chem. 2011 Apr;46(4):1103-16. doi: 10.1016/j.ejmech.2011.01.025. Epub 2011 Jan 21. Eur J Med Chem. 2011. PMID: 21316127 Free PMC article.

6

Mapping pilicide anti-virulence effect in Escherichia coli, a comprehensive structure-activity study.

Chorell E, Pinkner JS, Bengtsson C, Banchelin TS, Edvinsson S, Linusson A, Hultgren SJ, Almqvist F. Chorell E, et al. Among authors: almqvist f. Bioorg Med Chem. 2012 May 1;20(9):3128-42. doi: 10.1016/j.bmc.2012.01.048. Epub 2012 Feb 4. Bioorg Med Chem. 2012. PMID: 22464688 Free PMC article.

7

Design, synthesis and evaluation of triazole functionalized ring-fused 2-pyridones as antibacterial agents.

Bengtsson C, Lindgren AE, Uvell H, Almqvist F. Bengtsson C, et al. Among authors: almqvist f. Eur J Med Chem. 2012 Aug;54:637-46. doi: 10.1016/j.ejmech.2012.06.018. Epub 2012 Jun 18. Eur J Med Chem. 2012. PMID: 22749393 Free article.

8

Synthesis of fluorescent ring-fused 2-pyridone peptidomimetics.

Krishnan KS, Bengtsson C, Good JA, Mirkhanov S, Chorell E, Johansson LB, Almqvist F. Krishnan KS, et al. Among authors: almqvist f. J Org Chem. 2013 Dec 6;78(23):12207-13. doi: 10.1021/jo401844y. Epub 2013 Nov 14. J Org Chem. 2013. PMID: 24161000

9

Adhesive fiber stratification in uropathogenic Escherichia coli biofilms unveils oxygen-mediated control of type 1 pili.

Floyd KA, Moore JL, Eberly AR, Good JA, Shaffer CL, Zaver H, Almqvist F, Skaar EP, Caprioli RM, Hadjifrangiskou M. Floyd KA, et al. Among authors: almqvist f. PLoS Pathog. 2015 Mar 4;11(3):e1004697. doi: 10.1371/journal.ppat.1004697. eCollection 2015 Mar. PLoS Pathog. 2015. PMID: 25738819 Free PMC article.

10

Thiazolino 2-Pyridone Amide Inhibitors of Chlamydia trachomatis Infectivity.

Good JA, Silver J, Núñez-Otero C, Bahnan W, Krishnan KS, Salin O, Engström P, Svensson R, Artursson P, Gylfe Å, Bergström S, Almqvist F. Good JA, et al. Among authors: almqvist f. J Med Chem. 2016 Mar 10;59(5):2094-108. doi: 10.1021/acs.jmedchem.5b01759. Epub 2016 Feb 22. J Med Chem. 2016. PMID: 26849778

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