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Redirecting raltitrexed from cancer cell thymidylate synthase to Mycobacterium tuberculosis phosphopantetheinyl transferase.
Sci Adv. 2024 Mar 15;10(11):eadj6406. doi: 10.1126/sciadv.adj6406. Epub 2024 Mar 15.
Sci Adv. 2024.
PMID: 38489355
Free PMC article.
Mycobacterium tuberculosis PptT Inhibitors Based on Heterocyclic Replacements of Amidinoureas.
Ottavi S, Li K, Cacioppo JG, Perkowski AJ, Ramesh R, Gold BS, Ling Y, Roberts J, Singh A, Zhang D, Mosior J, Goullieux L, Roubert C, Bacqué E, Sacchettini JC, Nathan CF, Aubé J.
Ottavi S, et al. Among authors: mosior j.
ACS Med Chem Lett. 2023 Jun 26;14(7):970-976. doi: 10.1021/acsmedchemlett.3c00162. eCollection 2023 Jul 13.
ACS Med Chem Lett. 2023.
PMID: 37465309
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In Vitro and In Vivo Inhibition of the Mycobacterium tuberculosis Phosphopantetheinyl Transferase PptT by Amidinoureas.
Ottavi S, Scarry SM, Mosior J, Ling Y, Roberts J, Singh A, Zhang D, Goullieux L, Roubert C, Bacqué E, Lagiakos HR, Vendome J, Moraca F, Li K, Perkowski AJ, Ramesh R, Bowler MM, Tracy W, Feher VA, Sacchettini JC, Gold BS, Nathan CF, Aubé J.
Ottavi S, et al. Among authors: mosior j.
J Med Chem. 2022 Feb 10;65(3):1996-2022. doi: 10.1021/acs.jmedchem.1c01565. Epub 2022 Jan 19.
J Med Chem. 2022.
PMID: 35044775
Free PMC article.
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Characterization of Phosphopantetheinyl Hydrolase from Mycobacterium tuberculosis.
Pandey S, Singh A, Yang G, d'Andrea FB, Jiang X, Hartman TE, Mosior JW, Bourland R, Gold B, Roberts J, Geiger A, Tang S, Rhee K, Ouerfelli O, Sacchettini JC, Nathan CF, Burns-Huang K.
Pandey S, et al. Among authors: mosior jw.
Microbiol Spectr. 2021 Oct 31;9(2):e0092821. doi: 10.1128/Spectrum.00928-21. Epub 2021 Sep 22.
Microbiol Spectr. 2021.
PMID: 34550010
Free PMC article.
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Structural insights into phosphopantetheinyl hydrolase PptH from Mycobacterium tuberculosis.
Mosior J, Bourland R, Soma S, Nathan C, Sacchettini J.
Mosior J, et al.
Protein Sci. 2020 Mar;29(3):744-757. doi: 10.1002/pro.3813. Epub 2020 Jan 20.
Protein Sci. 2020.
PMID: 31886928
Free PMC article.
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Opposing reactions in coenzyme A metabolism sensitize Mycobacterium tuberculosis to enzyme inhibition.
Ballinger E, Mosior J, Hartman T, Burns-Huang K, Gold B, Morris R, Goullieux L, Blanc I, Vaubourgeix J, Lagrange S, Fraisse L, Sans S, Couturier C, Bacqué E, Rhee K, Scarry SM, Aubé J, Yang G, Ouerfelli O, Schnappinger D, Ioerger TR, Engelhart CA, McConnell JA, McAulay K, Fay A, Roubert C, Sacchettini J, Nathan C.
Ballinger E, et al. Among authors: mosior j.
Science. 2019 Feb 1;363(6426):eaau8959. doi: 10.1126/science.aau8959.
Science. 2019.
PMID: 30705156
Free PMC article.
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Unlocking Endosomal Entrapment with Supercharged Arginine-Rich Peptides.
Najjar K, Erazo-Oliveras A, Mosior JW, Whitlock MJ, Rostane I, Cinclair JM, Pellois JP.
Najjar K, et al. Among authors: mosior jw.
Bioconjug Chem. 2017 Dec 20;28(12):2932-2941. doi: 10.1021/acs.bioconjchem.7b00560. Epub 2017 Nov 13.
Bioconjug Chem. 2017.
PMID: 29065262
Free PMC article.
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An active role for the ribosome in determining the fate of oxidized mRNA.
Simms CL, Hudson BH, Mosior JW, Rangwala AS, Zaher HS.
Simms CL, et al. Among authors: mosior jw.
Cell Rep. 2014 Nov 20;9(4):1256-64. doi: 10.1016/j.celrep.2014.10.042. Epub 2014 Nov 13.
Cell Rep. 2014.
PMID: 25456128
Free PMC article.
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