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Page 1
BACE-1 Inhibitors Targeting Alzheimer's Disease.
Monteiro KLC, Dos Santos Alcântara MG, Freire NML, Brandão EM, do Nascimento VL, Dos Santos Viana LM, de Aquino TM, da Silva-Júnior EF. Monteiro KLC, et al. Among authors: de aquino tm. Curr Alzheimer Res. 2023;20(3):131-148. doi: 10.2174/1567205020666230612155953. Curr Alzheimer Res. 2023. PMID: 37309767 Review.
2-Amino-thiophene derivatives present antileishmanial activity mediated by apoptosis and immunomodulation in vitro.
Rodrigues KA, Dias CN, Néris PL, Rocha Jda C, Scotti MT, Scotti L, Mascarenhas SR, Veras RC, de Medeiros IA, Keesen Tde S, de Oliveira TB, de Lima Mdo C, Balliano TL, de Aquino TM, de Moura RO, Mendonça Junior FJ, de Oliveira MR. Rodrigues KA, et al. Among authors: de moura ro, de aquino tm, de lima mdo c, de oliveira mr, de oliveira tb, de medeiros ia. Eur J Med Chem. 2015 Dec 1;106:1-14. doi: 10.1016/j.ejmech.2015.10.011. Epub 2015 Oct 17. Eur J Med Chem. 2015. PMID: 26513640
Synthesis and evaluation of anti-Toxoplasma gondii and antimicrobial activities of thiosemicarbazides, 4-thiazolidinones and 1,3,4-thiadiazoles.
Liesen AP, de Aquino TM, Carvalho CS, Lima VT, de Araújo JM, de Lima JG, de Faria AR, de Melo EJ, Alves AJ, Alves EW, Alves AQ, Góes AJ. Liesen AP, et al. Among authors: de melo ej, de aquino tm, de araujo jm, de lima jg, de faria ar. Eur J Med Chem. 2010 Sep;45(9):3685-91. doi: 10.1016/j.ejmech.2010.05.017. Epub 2010 May 31. Eur J Med Chem. 2010. PMID: 20541294
Antileishmanial activity of new thiophene-indole hybrids: Design, synthesis, biological and cytotoxic evaluation, and chemometric studies.
Félix MB, de Souza ER, de Lima MDCA, Frade DKG, Serafim VL, Rodrigues KADF, Néris PLDN, Ribeiro FF, Scotti L, Scotti MT, de Aquino TM, Mendonça Junior FJB, de Oliveira MR. Félix MB, et al. Among authors: de aquino tm, de oliveira mr, de souza er, de lima mdca. Bioorg Med Chem. 2016 Sep 15;24(18):3972-3977. doi: 10.1016/j.bmc.2016.04.057. Epub 2016 Apr 26. Bioorg Med Chem. 2016. PMID: 27515718 Free article.
Dynamic Simulation, Docking and DFT Studies Applied to a Set of Anti-Acetylcholinesterase Inhibitors in the enzyme β-Secretase (BACE-1): An Important Therapeutic Target in Alzheimer`s disease.
Silva-Junior EF, Barcellos Franca PH, Quintans-Junior LJ, Mendonca-Junior FJB, Scotti L, Scotti MT, de Aquino TM, de Araujo-Junior JX. Silva-Junior EF, et al. Among authors: de araujo junior jx, de aquino tm. Curr Comput Aided Drug Des. 2017 Nov 10;13(4):266-274. doi: 10.2174/1573409913666170406150905. Curr Comput Aided Drug Des. 2017. PMID: 28382866
Molecular Docking Studies Applied to a Dataset of Cruzain Inhibitors.
da Silva-Junior EF, Barcellos Franca PH, Ribeiro FF, Bezerra Mendonca-Junior FJ, Scotti L, Scotti MT, de Aquino TM, de Araujo-Junior JX. da Silva-Junior EF, et al. Among authors: de araujo junior jx, de aquino tm. Curr Comput Aided Drug Des. 2018;14(1):68-78. doi: 10.2174/1573409913666170519112758. Curr Comput Aided Drug Des. 2018. PMID: 28523999
Aminoguanidine hydrazones (AGH's) as modulators of norfloxacin resistance in Staphylococcus aureus that overexpress NorA efflux pump.
Dantas N, de Aquino TM, de Araújo-Júnior JX, da Silva-Júnior E, Gomes EA, Gomes AAS, Siqueira-Júnior JP, Mendonça Junior FJB. Dantas N, et al. Among authors: de araujo junior jx, de aquino tm. Chem Biol Interact. 2018 Jan 25;280:8-14. doi: 10.1016/j.cbi.2017.12.009. Epub 2017 Dec 5. Chem Biol Interact. 2018. PMID: 29208359
Annonalide and derivatives: Semisynthesis, cytotoxic activities and studies on interaction of annonalide with DNA.
Marques RA, Gomes AOCV, de Brito MV, Dos Santos ALP, da Silva GS, de Lima LB, Nunes FM, de Mattos MC, de Oliveira FCE, do Ó Pessoa C, de Moraes MO, de Fátima Â, Franco LL, Silva MM, Dantas MDA, Santos JCC, Figueiredo IM, da Silva-Júnior EF, de Aquino TM, de Araújo-Júnior JX, de Oliveira MCF, Leslie Gunatilaka AA. Marques RA, et al. Among authors: de araujo junior jx, de aquino tm, de oliveira mcf, de lima lb, de mattos mc, de moraes mo, de fatima a, de oliveira fce, de brito mv. J Photochem Photobiol B. 2018 Feb;179:156-166. doi: 10.1016/j.jphotobiol.2018.01.016. Epub 2018 Feb 3. J Photochem Photobiol B. 2018. PMID: 29413989
Evidence for the involvement of TNF-α, IL-1β and IL-10 in the antinociceptive and anti-inflammatory effects of indole-3-guanylhydrazone hydrochloride, an aromatic aminoguanidine, in rodents.
Sandes SMS, Heimfarth L, Brito RG, Santos PL, Gouveia DN, Carvalho AMS, Quintans JSS, da Silva-Júnior EF, de Aquino TM, França PHB, de Araújo-Júnior JX, Albuquerque-Júnior RLC, Zengin G, Schmitt M, Bourguignon JJ, Quintans-Júnior LJ. Sandes SMS, et al. Among authors: de araujo junior jx, de aquino tm. Chem Biol Interact. 2018 Apr 25;286:1-10. doi: 10.1016/j.cbi.2018.02.026. Epub 2018 Feb 27. Chem Biol Interact. 2018. PMID: 29499192
Highly functionalized piperidines: Free radical scavenging, anticancer activity, DNA interaction and correlation with biological activity.
Das S, da Silva CJ, Silva MM, Dantas MDA, de Fátima Â, Góis Ruiz ALT, da Silva CM, de Carvalho JE, Santos JCC, Figueiredo IM, da Silva-Júnior EF, de Aquino TM, de Araújo-Júnior JX, Brahmachari G, Modolo LV. Das S, et al. Among authors: de araujo junior jx, de aquino tm, de fatima a, de carvalho je. J Adv Res. 2017 Oct 31;9:51-61. doi: 10.1016/j.jare.2017.10.010. eCollection 2018 Jan. J Adv Res. 2017. PMID: 30046486 Free PMC article.
41 results