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In vitro activity, ultrastructural analysis and in silico pharmacokinetic properties (ADMET) of thiazole compounds against adult worms of Schistosoma mansoni.
Acta Trop. 2023 Sep;245:106965. doi: 10.1016/j.actatropica.2023.106965. Epub 2023 Jun 7.
Acta Trop. 2023.
PMID: 37295486
Synthesis of 4-(4-chlorophenyl)thiazole compounds: in silico and in vitro evaluations as leishmanicidal and trypanocidal agents.
Cruz Filho IJD, Oliveira JF, Santos ACS, Pereira VRA, Lima MCA.
Cruz Filho IJD, et al.
An Acad Bras Cienc. 2023 May 1;95(1):e20220538. doi: 10.1590/0001-3765202320220538. eCollection 2023.
An Acad Bras Cienc. 2023.
PMID: 37132749
Free article.
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Plumbagin: A Promising In Vivo Antiparasitic Candidate against Schistosoma mansoni and In Silico Pharmacokinetic Properties (ADMET).
Silva LMN, França WWM, Santos VHB, Souza RAF, Silva AM, Diniz EGM, Aguiar TWA, Rocha JVR, Souza MAA, Nascimento WRC, Lima Neto RG, Cruz Filho IJ, Ximenes ECPA, Araújo HDA, Aires AL, Albuquerque MCPA.
Silva LMN, et al.
Biomedicines. 2023 Aug 22;11(9):2340. doi: 10.3390/biomedicines11092340.
Biomedicines. 2023.
PMID: 37760782
Free PMC article.
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In silico ADMET prediction, evaluation of cytotoxicity in mouse splenocytes and preliminary evaluation of in vitro antimalarial activity of 4-(4-chlorophenyl)thiazole compounds.
Silva BRMGD, Bezerra Júnior NDS, Oliveira JF, Duarte DMFA, Marques DSC, Nogueira F, Lima MCA, Cruz Filho IJD.
Silva BRMGD, et al. Among authors: cruz filho ijd.
An Acad Bras Cienc. 2023 Dec 4;95(suppl 2):e20230566. doi: 10.1590/0001-3765202320230566. eCollection 2023.
An Acad Bras Cienc. 2023.
PMID: 38055446
Free article.
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Alkaline lignins from Morinda citrifolia leaves are potential immunomodulatory, antitumor, and antimicrobial agents.
Cruz Filho IJ, Reis DP, Nascimento PHB, Marques DSC, Lima MCA.
Cruz Filho IJ, et al.
An Acad Bras Cienc. 2023 Dec 1;95(suppl 2):e20221026. doi: 10.1590/0001-3765202320221026. eCollection 2023.
An Acad Bras Cienc. 2023.
PMID: 38055562
Free article.
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Saline extract from Malpighia emarginata DC leaves showed higher polyphenol presence, antioxidant and antifungal activity and promoted cell proliferation in mice splenocytes.
Barros BRS, Barboza BR, Ramos BA, Moura MC, Coelho LCBB, Napoleão TH, Correia MTS, Paiva PMG, Cruz Filho IJD, Silva TDD, Lima CSA, Melo CML.
Barros BRS, et al. Among authors: cruz filho ijd.
An Acad Bras Cienc. 2019;91(1):e20190916. doi: 10.1590/0001-3765201920180358. Epub 2019 Apr 8.
An Acad Bras Cienc. 2019.
PMID: 30994765
Free article.
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