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ACW-02 an Acridine Triazolidine Derivative Presents Antileishmanial Activity Mediated by DNA Interaction and Immunomodulation.
Pharmaceuticals (Basel). 2023 Jan 29;16(2):204. doi: 10.3390/ph16020204.
Pharmaceuticals (Basel). 2023.
PMID: 37259353
Free PMC article.
Targeting SmCB1: Perspectives and Insights to Design Antischistosomal Drugs.
Dos Santos Nascimento IJ, Albino SL, da Silva Menezes KJ, de Azevedo Teotônio Cavalcanti M, de Oliveira MS, Mali SN, de Moura RO.
Dos Santos Nascimento IJ, et al.
Curr Med Chem. 2024;31(16):2264-2284. doi: 10.2174/0109298673255826231011114249.
Curr Med Chem. 2024.
PMID: 37921174
Review.
Item in Clipboard
Overview of the New Bioactive Heterocycles as Targeting Topoisomerase Inhibitors Useful Against Colon Cancer.
Santos MB, de Azevedo Teotônio Cavalcanti M, de Medeiros E Silva YMS, Dos Santos Nascimento IJ, de Moura RO.
Santos MB, et al.
Anticancer Agents Med Chem. 2024;24(4):236-262. doi: 10.2174/0118715206269722231121173311.
Anticancer Agents Med Chem. 2024.
PMID: 38038012
Review.
Item in Clipboard
Insights to Design New Drugs against Human African Trypanosomiasis Targeting Rhodesain using Covalent Docking, Molecular Dynamics Simulations, and MM-PBSA Calculations.
Nascimento IJDS, Santos MB, Marinho WPJ, Moura RO.
Nascimento IJDS, et al.
Curr Comput Aided Drug Des. 2024 Jan 19. doi: 10.2174/0115734099274797231205055827. Online ahead of print.
Curr Comput Aided Drug Des. 2024.
PMID: 38310575
Item in Clipboard
Exploring N-myristoyltransferase as a promising drug target against parasitic neglected tropical diseases.
Nascimento IJDS, Cavalcanti MAT, de Moura RO.
Nascimento IJDS, et al.
Eur J Med Chem. 2023 Oct 5;258:115550. doi: 10.1016/j.ejmech.2023.115550. Epub 2023 Jun 8.
Eur J Med Chem. 2023.
PMID: 37336067
Review.
Item in Clipboard
The new psychoactive substances 25H-NBOMe and 25H-NBOH induce abnormal development in the zebrafish embryo and interact in the DNA major groove.
de Barros WA, Nunes CDS, Souza JADCR, Nascimento IJDS, Figueiredo IM, de Aquino TM, Vieira L, Farias D, Santos JCC, de Fátima Â.
de Barros WA, et al. Among authors: nascimento ijds.
Curr Res Toxicol. 2021 Nov 22;2:386-398. doi: 10.1016/j.crtox.2021.11.002. eCollection 2021.
Curr Res Toxicol. 2021.
PMID: 34888530
Free PMC article.
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Insights on Dengue and Zika NS5 RNA-dependent RNA polymerase (RdRp) inhibitors.
Nascimento IJDS, Santos-Júnior PFDS, Aquino TM, Araújo-Júnior JX, Silva-Júnior EFD.
Nascimento IJDS, et al.
Eur J Med Chem. 2021 Nov 15;224:113698. doi: 10.1016/j.ejmech.2021.113698. Epub 2021 Jul 13.
Eur J Med Chem. 2021.
PMID: 34274831
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