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Evaluation of phthalazinone phosphodiesterase inhibitors with improved activity and selectivity against Trypanosoma cruzi.
De Araújo JS, da Silva PB, Batista MM, Peres RB, Cardoso-Santos C, Kalejaiye TD, Munday JC, De Heuvel E, Sterk GJ, Augustyns K, Salado IG, Matheeussen A, De Esch I, De Koning HP, Leurs R, Maes L, Soeiro MNC. De Araújo JS, et al. Among authors: de koning hp, de heuvel e, de esch i. J Antimicrob Chemother. 2020 Apr 1;75(4):958-967. doi: 10.1093/jac/dkz516. J Antimicrob Chemother. 2020. PMID: 31860098
Efficacy of Novel Pyrazolone Phosphodiesterase Inhibitors in Experimental Mouse Models of Trypanosoma cruzi.
de Araújo JS, França da Silva C, Batista DDGJ, Nefertiti A, Fiuza LFA, Fonseca-Berzal CR, Bernardino da Silva P, Batista MM, Sijm M, Kalejaiye TD, de Koning HP, Maes L, Sterk GJ, Leurs R, Soeiro MNC. de Araújo JS, et al. Among authors: de koning hp. Antimicrob Agents Chemother. 2020 Aug 20;64(9):e00414-20. doi: 10.1128/AAC.00414-20. Print 2020 Aug 20. Antimicrob Agents Chemother. 2020. PMID: 32601163 Free PMC article.
Positively selected modifications in the pore of TbAQP2 allow pentamidine to enter Trypanosoma brucei.
Alghamdi AH, Munday JC, Campagnaro GD, Gurvic D, Svensson F, Okpara CE, Kumar A, Quintana J, Martin Abril ME, Milić P, Watson L, Paape D, Settimo L, Dimitriou A, Wielinska J, Smart G, Anderson LF, Woodley CM, Kelly SPY, Ibrahim HM, Hulpia F, Al-Salabi MI, Eze AA, Sprenger T, Teka IA, Gudin S, Weyand S, Field M, Dardonville C, Tidwell RR, Carrington M, O'Neill P, Boykin DW, Zachariae U, De Koning HP. Alghamdi AH, et al. Among authors: de koning hp. Elife. 2020 Aug 11;9:e56416. doi: 10.7554/eLife.56416. Elife. 2020. PMID: 32762841 Free PMC article.
Tetrahydrophthalazinone Inhibitor of Phosphodiesterase with In Vitro Activity against Intracellular Trypanosomatids.
de Araújo JS, Peres RB, Bernardino da Silva P, Batista MM, Sterk GJ, Maes L, Caljon G, Leurs R, de Koning HP, Kalejaiye TD, Soeiro MNC. de Araújo JS, et al. Among authors: de koning hp. Antimicrob Agents Chemother. 2021 Feb 17;65(3):e00960-20. doi: 10.1128/AAC.00960-20. Print 2021 Feb 17. Antimicrob Agents Chemother. 2021. PMID: 33361300 Free PMC article.
Diamidines for human African trypanosomiasis.
Paine MF, Wang MZ, Generaux CN, Boykin DW, Wilson WD, De Koning HP, Olson CA, Pohlig G, Burri C, Brun R, Murilla GA, Thuita JK, Barrett MP, Tidwell RR. Paine MF, et al. Among authors: de koning hp. Curr Opin Investig Drugs. 2010 Aug;11(8):876-83. Curr Opin Investig Drugs. 2010. PMID: 20721830 Review.
Imidazole Derivatives as Promising Agents for the Treatment of Chagas Disease.
de Araújo JS, García-Rubia A, Sebastián-Pérez V, Kalejaiye TD, Bernardino da Silva P, Fonseca-Berzal CR, Maes L, De Koning HP, Soeiro MNC, Gil C. de Araújo JS, et al. Among authors: de koning hp. Antimicrob Agents Chemother. 2019 Mar 27;63(4):e02156-18. doi: 10.1128/AAC.02156-18. Print 2019 Apr. Antimicrob Agents Chemother. 2019. PMID: 30670432 Free PMC article.
180 results