Xia G - Search Results

1

Discovery of novel triazoles containing benzyloxy phenyl isoxazole side chain with potent and broad-spectrum antifungal activity.

Chi X, Xie F, Li L, Hao Y, Wu H, Li X, Xia G, Yan L, Zhang D, Jiang Y, Ni T. Chi X, et al. Among authors: xia g. Bioorg Chem. 2023 Aug;137:106572. doi: 10.1016/j.bioorg.2023.106572. Epub 2023 Apr 28. Bioorg Chem. 2023. PMID: 37156136

2

Potent and novel 11β-HSD1 inhibitors identified from shape and docking based virtual screening.

Xia G, Xue M, Liu L, Yu J, Liu H, Li P, Wang J, Li Y, Xiong B, Shen J. Xia G, et al. Bioorg Med Chem Lett. 2011 Oct 1;21(19):5739-44. doi: 10.1016/j.bmcl.2011.08.019. Epub 2011 Aug 8. Bioorg Med Chem Lett. 2011. PMID: 21873057

3

Discovery and optimization of a series of imidazo[4,5-b]pyrazine derivatives as highly potent and exquisitely selective inhibitors of the mesenchymal-epithelial transition factor (c-Met) protein kinase.

Zhao F, Zhang J, Zhang L, Hao Y, Shi C, Xia G, Yu J, Liu Y. Zhao F, et al. Among authors: xia g. Bioorg Med Chem. 2016 Sep 15;24(18):4281-4290. doi: 10.1016/j.bmc.2016.07.019. Epub 2016 Jul 12. Bioorg Med Chem. 2016. PMID: 27448775

4

Erratum to "Discovery and optimization of a series of imidazo[4,5-b]pyrazine derivatives as highly potent and exquisitely selective inhibitors of the mesenchymal-epithelial transition factor (c-Met) protein kinase" [Bioorg. Med. Chem. 24 (2016) 4281-4290].

Zhao F, Zhang J, Zhang L, Hao Y, Shi C, Xia G, Yu J, Liu Y. Zhao F, et al. Among authors: xia g. Bioorg Med Chem. 2017 May 15;25(10):2811-2812. doi: 10.1016/j.bmc.2017.03.042. Epub 2017 Apr 5. Bioorg Med Chem. 2017. PMID: 28389111 No abstract available.

5

Design, synthesis, and pharmacological evaluation of quinazoline derivatives as novel and potent pan-JAK inhibitors.

Xiang J, Wang Y, Wang W, Yu J, Zheng L, Hong Y, Shi L, Zhang C, Chen N, Xu J, Gong X, Zhang Z, Cui H, Zhou Q, Zhang D, Liu Y, Ke Y, Shen J, Xia G, Bai X. Xiang J, et al. Among authors: xia g. Bioorg Chem. 2023 Nov;140:106765. doi: 10.1016/j.bioorg.2023.106765. Epub 2023 Aug 7. Bioorg Chem. 2023. PMID: 37582330

6

Synthesis and phosphodiesterase 5 inhibitory activity of novel pyrido[1,2-e]purin-4(3H)-one derivatives.

Xia G, Li J, Peng A, Lai S, Zhang S, Shen J, Liu Z, Chen X, Ji R. Xia G, et al. Bioorg Med Chem Lett. 2005 Jun 2;15(11):2790-4. doi: 10.1016/j.bmcl.2005.03.102. Bioorg Med Chem Lett. 2005. PMID: 15878277

7

Discovery of novel sulfonamides as potent and selective inhibitors against human and mouse 11β-hydroxysteroid dehydrogenase type 1.

Xia G, Liu L, Xue M, Liu H, Yu J, Li P, Chen Q, Xiong B, Liu X, Shen J. Xia G, et al. Mol Cell Endocrinol. 2012 Jul 6;358(1):46-52. doi: 10.1016/j.mce.2012.02.017. Epub 2012 Mar 3. Mol Cell Endocrinol. 2012. PMID: 22410288

8

Design, synthesis and SAR of piperidyl-oxadiazoles as 11β-hydroxysteroid dehydrogenase 1 inhibitors.

Xia G, You X, Liu L, Liu H, Wang J, Shi Y, Li P, Xiong B, Liu X, Shen J. Xia G, et al. Eur J Med Chem. 2013 Apr;62:1-10. doi: 10.1016/j.ejmech.2012.12.059. Epub 2013 Jan 10. Eur J Med Chem. 2013. PMID: 23353742

9

Identification of 3-substituted-6-(1-(1H-[1,2,3]triazolo[4,5-b]pyrazin-1-yl)ethyl)quinoline derivatives as highly potent and selective mesenchymal-epithelial transition factor (c-Met) inhibitors via metabolite profiling-based structural optimization.

Zhao F, Zhang LD, Hao Y, Chen N, Bai R, Wang YJ, Zhang CC, Li GS, Hao LJ, Shi C, Zhang J, Mao Y, Fan Y, Xia GX, Yu JX, Liu YJ. Zhao F, et al. Eur J Med Chem. 2017 Jul 7;134:147-158. doi: 10.1016/j.ejmech.2017.03.085. Epub 2017 Apr 4. Eur J Med Chem. 2017. PMID: 28411455

10

Discovery of 6-(2-(dimethylamino)ethyl)-N-(5-fluoro-4-(4-fluoro-1-isopropyl-2-methyl-1H-benzo[d]imidazole-6-yl)pyrimidin-2-yl)-5,6,7,8-tetrahydro-1,6-naphthyridin-2-amine as a highly potent cyclin-dependent kinase 4/6 inhibitor for treatment of cancer.

Shi C, Wang Q, Liao X, Ge H, Huo G, Zhang L, Chen N, Zhai X, Hong Y, Wang L, Han Y, Xiao W, Wang Z, Shi W, Mao Y, Yu J, Xia G, Liu Y. Shi C, et al. Among authors: xia g. Eur J Med Chem. 2019 Sep 15;178:352-364. doi: 10.1016/j.ejmech.2019.06.005. Epub 2019 Jun 4. Eur J Med Chem. 2019. PMID: 31200237

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