Wilkinson S - Search Results

1

Systematic study of 1,2,3-triazolyl sterols for the development of new drugs against parasitic Neglected Tropical Diseases.

Porta EOJ, Ballari MS, Carlucci R, Wilkinson S, Ma G, Tekwani BL, Labadie GR. Porta EOJ, et al. Among authors: wilkinson s. Eur J Med Chem. 2023 Jun 5;254:115378. doi: 10.1016/j.ejmech.2023.115378. Epub 2023 Apr 13. Eur J Med Chem. 2023. PMID: 37084599

2

Synthesis and antikinetoplastid activity of a series of N,N'-substituted diamines.

Caminos AP, Panozzo-Zenere EA, Wilkinson SR, Tekwani BL, Labadie GR. Caminos AP, et al. Bioorg Med Chem Lett. 2012 Feb 15;22(4):1712-5. doi: 10.1016/j.bmcl.2011.12.101. Epub 2011 Dec 28. Bioorg Med Chem Lett. 2012. PMID: 22248858

3

Novel nitro(triazole/imidazole)-based heteroarylamides/sulfonamides as potential antitrypanosomal agents.

Papadopoulou MV, Bloomer WD, Rosenzweig HS, Wilkinson SR, Kaiser M. Papadopoulou MV, et al. Among authors: wilkinson sr. Eur J Med Chem. 2014 Nov 24;87:79-88. doi: 10.1016/j.ejmech.2014.09.045. Epub 2014 Sep 16. Eur J Med Chem. 2014. PMID: 25240098

4

3-Nitrotriazole-based piperazides as potent antitrypanosomal agents.

Papadopoulou MV, Bloomer WD, Rosenzweig HS, O'Shea IP, Wilkinson SR, Kaiser M. Papadopoulou MV, et al. Among authors: wilkinson sr. Eur J Med Chem. 2015 Oct 20;103:325-34. doi: 10.1016/j.ejmech.2015.08.042. Epub 2015 Sep 4. Eur J Med Chem. 2015. PMID: 26363868

5

Antitrypanosomal activity of 5-nitro-2-aminothiazole-based compounds.

Papadopoulou MV, Bloomer WD, Rosenzweig HS, Wilkinson SR, Szular J, Kaiser M. Papadopoulou MV, et al. Among authors: wilkinson sr. Eur J Med Chem. 2016 Jul 19;117:179-86. doi: 10.1016/j.ejmech.2016.04.010. Epub 2016 Apr 8. Eur J Med Chem. 2016. PMID: 27092415 Free PMC article.

6

Nitrotriazole-based acetamides and propanamides with broad spectrum antitrypanosomal activity.

Papadopoulou MV, Bloomer WD, Rosenzweig HS, Wilkinson SR, Szular J, Kaiser M. Papadopoulou MV, et al. Among authors: wilkinson sr. Eur J Med Chem. 2016 Nov 10;123:895-904. doi: 10.1016/j.ejmech.2016.08.002. Epub 2016 Aug 9. Eur J Med Chem. 2016. PMID: 27543881 Free PMC article.

7

Trypanocidal drugs: mechanisms, resistance and new targets.

Wilkinson SR, Kelly JM. Wilkinson SR, et al. Expert Rev Mol Med. 2009 Oct 29;11:e31. doi: 10.1017/S1462399409001252. Expert Rev Mol Med. 2009. PMID: 19863838 Free article. Review.

8

Nifurtimox activation by trypanosomal type I nitroreductases generates cytotoxic nitrile metabolites.

Hall BS, Bot C, Wilkinson SR. Hall BS, et al. Among authors: wilkinson sr. J Biol Chem. 2011 Apr 15;286(15):13088-95. doi: 10.1074/jbc.M111.230847. Epub 2011 Feb 23. J Biol Chem. 2011. PMID: 21345801 Free PMC article.

9

An essential type I nitroreductase from Leishmania major can be used to activate leishmanicidal prodrugs.

Voak AA, Gobalakrishnapillai V, Seifert K, Balczo E, Hu L, Hall BS, Wilkinson SR. Voak AA, et al. Among authors: wilkinson sr. J Biol Chem. 2013 Oct 4;288(40):28466-76. doi: 10.1074/jbc.M113.494781. Epub 2013 Aug 14. J Biol Chem. 2013. PMID: 23946481 Free PMC article.

10

Discovery of potent nitrotriazole-based antitrypanosomal agents: In vitro and in vivo evaluation.

Papadopoulou MV, Bloomer WD, Rosenzweig HS, O'Shea IP, Wilkinson SR, Kaiser M, Chatelain E, Ioset JR. Papadopoulou MV, et al. Among authors: wilkinson sr. Bioorg Med Chem. 2015 Oct 1;23(19):6467-76. doi: 10.1016/j.bmc.2015.08.014. Epub 2015 Aug 24. Bioorg Med Chem. 2015. PMID: 26344593

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