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A Selective ALDH1A3 Inhibitor Impairs Mesothelioma 3-D Multicellular Spheroid Growth and Neutrophil Recruitment.
Int J Mol Sci. 2023 Apr 3;24(7):6689. doi: 10.3390/ijms24076689.
Int J Mol Sci. 2023.
PMID: 37047661
Free PMC article.
Progress in the Field of Aldehyde Dehydrogenase Inhibitors: Novel Imidazo[1,2-a]pyridines against the 1A Family.
Quattrini L, Gelardi ELM, Petrarolo G, Colombo G, Ferraris DM, Picarazzi F, Rizzi M, Garavaglia S, La Motta C.
Quattrini L, et al. Among authors: petrarolo g.
ACS Med Chem Lett. 2020 Mar 25;11(5):963-970. doi: 10.1021/acsmedchemlett.9b00686. eCollection 2020 May 14.
ACS Med Chem Lett. 2020.
PMID: 32435412
Free PMC article.
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Aldehyde Dehydrogenases and Prostate Cancer: Shedding Light on Isoform Distribution to Reveal Druggable Target.
Quattrini L, Sadiq M, Petrarolo G, Maitland NJ, Frame FM, Pors K, La Motta C.
Quattrini L, et al. Among authors: petrarolo g.
Biomedicines. 2020 Dec 4;8(12):569. doi: 10.3390/biomedicines8120569.
Biomedicines. 2020.
PMID: 33291762
Free PMC article.
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A Selective Competitive Inhibitor of Aldehyde Dehydrogenase 1A3 Hinders Cancer Cell Growth, Invasiveness and Stemness In Vitro.
Gelardi ELM, Colombo G, Picarazzi F, Ferraris DM, Mangione A, Petrarolo G, Aronica E, Rizzi M, Mori M, La Motta C, Garavaglia S.
Gelardi ELM, et al. Among authors: petrarolo g.
Cancers (Basel). 2021 Jan 19;13(2):356. doi: 10.3390/cancers13020356.
Cancers (Basel). 2021.
PMID: 33478031
Free PMC article.
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Identification of novel SIRT1 activators endowed with cardioprotective profile.
Flori L, Petrarolo G, Brogi S, La Motta C, Testai L, Calderone V.
Flori L, et al. Among authors: petrarolo g.
Eur J Pharm Sci. 2021 Oct 1;165:105930. doi: 10.1016/j.ejps.2021.105930. Epub 2021 Jul 12.
Eur J Pharm Sci. 2021.
PMID: 34265406
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Aurones: A Golden Resource for Active Compounds.
Mazziotti I, Petrarolo G, La Motta C.
Mazziotti I, et al. Among authors: petrarolo g.
Molecules. 2021 Dec 21;27(1):2. doi: 10.3390/molecules27010002.
Molecules. 2021.
PMID: 35011233
Free PMC article.
Review.
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Nature-Inspired O-Benzyl Oxime-Based Derivatives as New Dual-Acting Agents Targeting Aldose Reductase and Oxidative Stress.
Ciccone L, Petrarolo G, Barsuglia F, Fruchart-Gaillard C, Cassar Lajeunesse E, Adewumi AT, Soliman MES, La Motta C, Orlandini E, Nencetti S.
Ciccone L, et al. Among authors: petrarolo g.
Biomolecules. 2022 Mar 14;12(3):448. doi: 10.3390/biom12030448.
Biomolecules. 2022.
PMID: 35327641
Free PMC article.
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New Hybrid Compounds Incorporating Natural Products as Multifunctional Agents against Alzheimer's Disease.
Ciccone L, Camodeca C, Tonali N, Barlettani L, Rossello A, Fruchart Gaillard C, Kaffy J, Petrarolo G, La Motta C, Nencetti S, Orlandini E.
Ciccone L, et al. Among authors: petrarolo g.
Pharmaceutics. 2023 Sep 22;15(10):2369. doi: 10.3390/pharmaceutics15102369.
Pharmaceutics. 2023.
PMID: 37896129
Free PMC article.
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