Discovery of Orally Bioavailable Ligand Efficient Quinazolindiones as Potent and Selective Tankyrases Inhibitors.
Qin D, Lin X, Liu Z, Chen Y, Zhang Z, Wu C, Liu L, Pan Y, Laquerre S, Emery J, Fergusson J, Roland K, Keenan R, Oliff A, Kumar S, Cheung M, Su DS.
Qin D, et al. Among authors: liu z, liu l.
ACS Med Chem Lett. 2021 May 13;12(6):1005-1010. doi: 10.1021/acsmedchemlett.1c00160. eCollection 2021 Jun 10.
ACS Med Chem Lett. 2021.
PMID: 34141085
Free PMC article.