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Controlling Ibrutinib's Conformations about Its Heterobiaryl Axis to Increase BTK Selectivity.
ACS Med Chem Lett. 2023 Feb 14;14(3):305-311. doi: 10.1021/acsmedchemlett.2c00523. eCollection 2023 Mar 9.
ACS Med Chem Lett. 2023.
PMID: 36923918
Free PMC article.
Approaches toward Atropisomerically Stable and Conformationally Pure Diarylamines.
Vaidya SD, Heydari BS, Toenjes ST, Gustafson JL.
Vaidya SD, et al. Among authors: heydari bs.
J Org Chem. 2022 May 20;87(10):6760-6768. doi: 10.1021/acs.joc.2c00451. Epub 2022 Apr 29.
J Org Chem. 2022.
PMID: 35486501
Free PMC article.
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