Search Page
Save citations to file
Email citations
Send citations to clipboard
Add to Collections
Add to My Bibliography
Create a file for external citation management software
Your saved search
Your RSS Feed
Search Results
6 results
Filters applied: . Clear all
Results are displayed in a computed author sort order.
The Results By Year timeline is not available.
Page 1
APOBEC3A Catalytic Inactivity Mutation Induces Tertiary Structure Destabilization.
ACS Med Chem Lett. 2023 Feb 14;14(3):338-343. doi: 10.1021/acsmedchemlett.2c00517. eCollection 2023 Mar 9.
ACS Med Chem Lett. 2023.
PMID: 36923917
Free PMC article.
Differential Inhibition of APOBEC3 DNA-Mutator Isozymes by Fluoro- and Non-Fluoro-Substituted 2'-Deoxyzebularine Embedded in Single-Stranded DNA.
Kvach MV, Barzak FM, Harjes S, Schares HAM, Kurup HM, Jones KF, Sutton L, Donahue J, D'Aquila RT, Jameson GB, Harki DA, Krause KL, Harjes E, Filichev VV.
Kvach MV, et al.
Chembiochem. 2020 Apr 1;21(7):1028-1035. doi: 10.1002/cbic.201900505. Epub 2019 Dec 19.
Chembiochem. 2020.
PMID: 31633265
Free PMC article.
Item in Clipboard
Synthesis of Guaianolide Analogues with a Tunable α-Methylene-γ-lactam Electrophile and Correlating Bioactivity with Thiol Reactivity.
Jackson PA, Schares HAM, Jones KFM, Widen JC, Dempe DP, Grillet F, Cuellar ME, Walters MA, Harki DA, Brummond KM.
Jackson PA, et al. Among authors: jones kfm.
J Med Chem. 2020 Dec 10;63(23):14951-14978. doi: 10.1021/acs.jmedchem.0c01464. Epub 2020 Nov 17.
J Med Chem. 2020.
PMID: 33201697
Free PMC article.
Item in Clipboard
Function-Oriented and Modular (+/-)-cis-Pseudoguaianolide Synthesis: Discovery of New Nrf2 Activators and NF-κB Inhibitors.
Emmetiere F, Ratnayake R, Schares HAM, Jones KFM, Bevan-Smith E, Luesch H, Harki DA, Grenning AJ.
Emmetiere F, et al. Among authors: jones kfm.
Chemistry. 2021 Mar 22;27(17):5564-5571. doi: 10.1002/chem.202100038. Epub 2021 Feb 26.
Chemistry. 2021.
PMID: 33502811
Free PMC article.
Item in Clipboard
The current toolbox for APOBEC drug discovery.
Grillo MJ, Jones KFM, Carpenter MA, Harris RS, Harki DA.
Grillo MJ, et al. Among authors: jones kfm.
Trends Pharmacol Sci. 2022 May;43(5):362-377. doi: 10.1016/j.tips.2022.02.007.
Trends Pharmacol Sci. 2022.
PMID: 35272863
Free PMC article.
Review.
Item in Clipboard
Development of Allosteric Small Molecule APOBEC3B Inhibitors from In Silico Screening.
Jones KFM, Demir Ö, Wyllie MK, Grillo MJ, Morris C, Hirakis SP, Kardile RD, Walters MA, Harris RS, Amaro RE, Harki DA.
Jones KFM, et al.
bioRxiv [Preprint]. 2024 Apr 25:2024.04.25.591187. doi: 10.1101/2024.04.25.591187.
bioRxiv. 2024.
PMID: 38712210
Free PMC article.
Preprint.
Item in Clipboard
Cite
Cite