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Page 1
Synthesis, characterization, antioxidant and antiparasitic activities new naphthyl-thiazole derivatives.
Santos NFN, Junior NDSB, de Oliveira JF, Duarte DMFA, Dos Santos Soares JC, Clara Marques DS, da Silva Santos AC, Nogueira F, Alves Pereira VR, Alves de Lima MC, da Cruz Filho IJ. Santos NFN, et al. Among authors: de oliveira jf. Exp Parasitol. 2023 May;248:108498. doi: 10.1016/j.exppara.2023.108498. Epub 2023 Mar 11. Exp Parasitol. 2023. PMID: 36907541
Novel indol-3-yl-thiosemicarbazone derivatives: Obtaining, evaluation of in vitro leishmanicidal activity and ultrastructural studies.
da Silva PR, de Oliveira JF, da Silva AL, Queiroz CM, Feitosa APS, Duarte DMFA, da Silva AC, de Castro MCAB, Pereira VRA, da Silva RMF, Alves LC, Dos Santos FAB, de Lima MDCA. da Silva PR, et al. Among authors: de castro mcab, de oliveira jf, de lima mdca. Chem Biol Interact. 2020 Jan 5;315:108899. doi: 10.1016/j.cbi.2019.108899. Epub 2019 Nov 15. Chem Biol Interact. 2020. PMID: 31738906
Anti-inflammatory activity of novel thiosemicarbazone compounds indole-based as COX inhibitors.
Jacob ÍTT, Gomes FOS, de Miranda MDS, de Almeida SMV, da Cruz-Filho IJ, Peixoto CA, da Silva TG, Moreira DRM, de Melo CML, de Oliveira JF, de Lima MCA. Jacob ÍTT, et al. Among authors: de miranda mds, de almeida smv, de melo cml, de lima mca, de oliveira jf. Pharmacol Rep. 2021 Jun;73(3):907-925. doi: 10.1007/s43440-021-00221-7. Epub 2021 Feb 15. Pharmacol Rep. 2021. PMID: 33590474
Neurolocomotor Behavior and Oxidative Stress Markers of Thiazole and Thiazolidinedione Derivatives against Nauphoeta cinerea.
Pereira PS, Costa AR, de Oliveira TJS, Oliveira CVB, de Lima MDCA, de Oliveira JF, Kim B, Coutinho HDM, Duarte AE, Kamdem JP, da Silva TG. Pereira PS, et al. Among authors: de oliveira tjs, oliveira cvb, de lima mdca, de oliveira jf. Antioxidants (Basel). 2022 Feb 18;11(2):420. doi: 10.3390/antiox11020420. Antioxidants (Basel). 2022. PMID: 35204302 Free PMC article.
Synthesis, in vitro schistosomicidal activity and ultrastructural alterations caused by thiosemicarbazones and thiazolidinones against juvenile and adult Schistosoma mansoni worms (Sambon, 1907).
Tavares da Rocha RE, de Almeida Júnior ASA, Júnior NCP, do Nascimento AV, Leite NMS, de Oliveira JF, Alves de Lima MDC, Feitosa APS, Bezerra de Mélo ME, Brayner FA, Alves LC. Tavares da Rocha RE, et al. Among authors: de almeida junior asa, de oliveira jf. Mol Biochem Parasitol. 2022 Nov;252:111520. doi: 10.1016/j.molbiopara.2022.111520. Epub 2022 Sep 16. Mol Biochem Parasitol. 2022. PMID: 36122704 Free article.
In vitro activity, ultrastructural studies and in silico pharmacokinetic properties of indol-3-yl-thiosemicarbazones derivatives and analogues against juvenile and adult worms of S. mansoni.
de Almeida Júnior ASA, de Oliveira JF, da Silva AL, da Rocha RET, Junior NCP, Gouveia ALA, da Silva RMF, de Azevedo Albuquerque MCP, Brayner FA, Alves LC, do Carmo Alves de Lima M. de Almeida Júnior ASA, et al. Among authors: de azevedo albuquerque mcp, de oliveira jf. Eur J Pharm Sci. 2019 Oct 1;138:104985. doi: 10.1016/j.ejps.2019.104985. Epub 2019 Jul 5. Eur J Pharm Sci. 2019. PMID: 31283945
Thiazolidinedione and thiazole derivatives potentiate norfloxacin activity against NorA efflux pump over expression in Staphylococcus aureus 1199B strains.
Pereira PS, Lima MDCA, Neto PPM, Oliveira-Tintino CDM, Tintino SR, Menezes IRA, de Oliveira JF, Marchand P, Coutinho HDM, Rodrigues MDD, da Silva TG. Pereira PS, et al. Among authors: oliveira tintino cdm, de oliveira jf. Bioorg Med Chem. 2019 Sep 1;27(17):3797-3804. doi: 10.1016/j.bmc.2019.07.006. Epub 2019 Jul 4. Bioorg Med Chem. 2019. PMID: 31320212 Free article.
Novel indole-thiazole and indole-thiazolidinone derivatives as DNA groove binders.
Alves JEF, de Oliveira JF, de Lima Souza TRC, de Moura RO, de Carvalho Júnior LB, Alves de Lima MDC, de Almeida SMV. Alves JEF, et al. Among authors: de almeida smv, de moura ro, de carvalho junior lb, de lima souza trc, de oliveira jf. Int J Biol Macromol. 2021 Feb 15;170:622-635. doi: 10.1016/j.ijbiomac.2020.12.153. Epub 2021 Jan 5. Int J Biol Macromol. 2021. PMID: 33359805
Study of nitrogen heterocycles as DNA/HSA binder, topoisomerase inhibitors and toxicological safety.
Dos Santos JC, Alves JEF, de Azevedo RDS, de Lima ML, de Oliveira Silva MR, da Silva JG, da Silva JM, de Carvalho Correia AC, do Carmo Alves de Lima M, de Oliveira JF, de Moura RO, de Almeida SMV. Dos Santos JC, et al. Among authors: de oliveira jf. Int J Biol Macromol. 2024 Jan;254(Pt 3):127651. doi: 10.1016/j.ijbiomac.2023.127651. Epub 2023 Nov 8. Int J Biol Macromol. 2024. PMID: 37949265
139 results