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New Triazine Derivatives as Serotonin 5-HT6 Receptor Ligands.
Molecules. 2023 Jan 22;28(3):1108. doi: 10.3390/molecules28031108.
Molecules. 2023.
PMID: 36770774
Free PMC article.
Design, synthesis and structure-activity relationships of novel phenylalanine-based amino acids as kainate receptors ligands.
Szymańska E, Chałupnik P, Szczepańska K, Cuñado Moral AM, Pickering DS, Nielsen B, Johansen TN, Kieć-Kononowicz K.
Szymańska E, et al. Among authors: chalupnik p.
Bioorg Med Chem Lett. 2016 Nov 15;26(22):5568-5572. doi: 10.1016/j.bmcl.2016.09.075. Epub 2016 Sep 30.
Bioorg Med Chem Lett. 2016.
PMID: 27765511
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Aryl- and heteroaryl-substituted phenylalanines as AMPA receptor ligands.
Szymańska E, Chałupnik P, Johansen TN, Nielsen B, Cuñado Moral AM, Pickering DS, Więckowska A, Kieć-Kononowicz K.
Szymańska E, et al. Among authors: chalupnik p.
Chem Biol Drug Des. 2017 Dec;90(6):1271-1281. doi: 10.1111/cbdd.13048. Epub 2017 Jul 18.
Chem Biol Drug Des. 2017.
PMID: 28636281
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Discovery of the First Highly Selective Antagonist of the GluK3 Kainate Receptor Subtype.
Chałupnik P, Vialko A, Pickering DS, Hinkkanen M, Donbosco S, Møller TC, Jensen AA, Nielsen B, Bay Y, Kristensen AS, Johansen TN, Łątka K, Bajda M, Szymańska E.
Chałupnik P, et al.
Int J Mol Sci. 2022 Aug 8;23(15):8797. doi: 10.3390/ijms23158797.
Int J Mol Sci. 2022.
PMID: 35955932
Free PMC article.
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Kainate Receptor Antagonists: Recent Advances and Therapeutic Perspective.
Chałupnik P, Szymańska E.
Chałupnik P, et al.
Int J Mol Sci. 2023 Jan 18;24(3):1908. doi: 10.3390/ijms24031908.
Int J Mol Sci. 2023.
PMID: 36768227
Free PMC article.
Review.
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Structure-Activity Relationship and Solubility Studies of N1-Substituted Quinoxaline-2,3-diones as Kainate Receptor Antagonists.
Chałupnik P, Vialko A, Pickering DS, Nielsen B, Bay Y, Skov Kristensen A, Hinkkanen M, Szczepańska K, Karcz T, Latacz G, Johansen TN, Szymańska E.
Chałupnik P, et al.
ChemMedChem. 2023 Sep 15;18(18):e202300278. doi: 10.1002/cmdc.202300278. Epub 2023 Jul 20.
ChemMedChem. 2023.
PMID: 37387321
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N-(7-(1H-Imidazol-1-yl)-2,3-dioxo-6-(trifluoromethyl)-3,4-dihydroquinoxalin-1(2H)-yl)benzamide, a New Kainate Receptor Selective Antagonist and Analgesic: Synthesis, X-ray Crystallography, Structure-Affinity Relationships, and in Vitro and in Vivo Pharmacology.
Møllerud S, Hansen RB, Pallesen J, Temperini P, Pasini D, Bornholt J, Nielsen B, Mamedova E, Chalupnik P, Paternain AV, Lerma J, Diaz-delCastillo M, Andreasen JT, Frydenvang K, Kastrup JS, Johansen TN, Pickering DS.
Møllerud S, et al. Among authors: chalupnik p.
ACS Chem Neurosci. 2019 Nov 20;10(11):4685-4695. doi: 10.1021/acschemneuro.9b00479. Epub 2019 Oct 31.
ACS Chem Neurosci. 2019.
PMID: 31622082
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Tritium and deuterium labelling of a kainate receptor antagonist and evaluation as a radioligand.
Chałupnik P, Marek A, Hovah MEL, Pickering DS, Temperini P, Donbosco S, Szymańska E, Johansen TN.
Chałupnik P, et al.
J Labelled Comp Radiopharm. 2024 Apr;67(4):120-130. doi: 10.1002/jlcr.4087. Epub 2024 Feb 8.
J Labelled Comp Radiopharm. 2024.
PMID: 38332677
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