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Page 1
Preclinical Studies and Drug Combination of Low-Cost Molecules for Chagas Disease.
Aguilera E, Sánchez C, Cruces ME, Dávila B, Minini L, Mosquillo F, Pérez-Díaz L, Serna E, Torres S, Schini A, Sanabria L, Vera de Bilbao NI, Yaluff G, Zolessi FR, Ceilas LF, Cerecetto H, Alvarez G. Aguilera E, et al. Among authors: vera de bilbao ni. Pharmaceuticals (Basel). 2022 Dec 23;16(1):20. doi: 10.3390/ph16010020. Pharmaceuticals (Basel). 2022. PMID: 36678516 Free PMC article.
Optimization of antitrypanosomatid agents: identification of nonmutagenic drug candidates with in vivo activity.
Álvarez G, Varela J, Márquez P, Gabay M, Arias Rivas CE, Cuchilla K, Echeverría GA, Piro OE, Chorilli M, Leal SM, Escobar P, Serna E, Torres S, Yaluff G, Vera de Bilbao NI, González M, Cerecetto H. Álvarez G, et al. Among authors: vera de bilbao ni. J Med Chem. 2014 May 22;57(10):3984-99. doi: 10.1021/jm500018m. Epub 2014 May 2. J Med Chem. 2014. PMID: 24749923
Identification of a new amide-containing thiazole as a drug candidate for treatment of Chagas' disease.
Álvarez G, Varela J, Cruces E, Fernández M, Gabay M, Leal SM, Escobar P, Sanabria L, Serna E, Torres S, Figueredo Thiel SJ, Yaluff G, Vera de Bilbao NI, Cerecetto H, González M. Álvarez G, et al. Among authors: vera de bilbao ni. Antimicrob Agents Chemother. 2015 Mar;59(3):1398-404. doi: 10.1128/AAC.03814-14. Epub 2014 Dec 15. Antimicrob Agents Chemother. 2015. PMID: 25512408 Free PMC article.
A Nature-Inspired Design Yields a New Class of Steroids Against Trypanosomatids.
Aguilera E, Perdomo C, Espindola A, Corvo I, Faral-Tello P, Robello C, Serna E, Benítez F, Riveros R, Torres S, Vera de Bilbao NI, Yaluff G, Alvarez G. Aguilera E, et al. Among authors: vera de bilbao ni. Molecules. 2019 Oct 22;24(20):3800. doi: 10.3390/molecules24203800. Molecules. 2019. PMID: 31652542 Free PMC article.
In vitro and in vivo antitrypanosomatid activity of 5-nitroindazoles.
Boiani L, Gerpe A, Arán VJ, Torres de Ortiz S, Serna E, Vera de Bilbao N, Sanabria L, Yaluff G, Nakayama H, Rojas de Arias A, Maya JD, Morello JA, Cerecetto H, González M. Boiani L, et al. Eur J Med Chem. 2009 Mar;44(3):1034-40. doi: 10.1016/j.ejmech.2008.06.024. Epub 2008 Jun 28. Eur J Med Chem. 2009. PMID: 18706738
Development of bis-thiazoles as inhibitors of triosephosphate isomerase from Trypanosoma cruzi. Identification of new non-mutagenic agents that are active in vivo.
Álvarez G, Martínez J, Varela J, Birriel E, Cruces E, Gabay M, Leal SM, Escobar P, Aguirre-López B, Cabrera N, Tuena de Gómez-Puyou M, Gómez Puyou A, Pérez-Montfort R, Yaluff G, Torres S, Serna E, Vera de Bilbao N, González M, Cerecetto H. Álvarez G, et al. Eur J Med Chem. 2015 Jul 15;100:246-56. doi: 10.1016/j.ejmech.2015.06.018. Epub 2015 Jun 12. Eur J Med Chem. 2015. PMID: 26094151
3-Trifluoromethylquinoxaline N,N'-dioxides as anti-trypanosomatid agents. Identification of optimal anti-T. cruzi agents and mechanism of action studies.
Benitez D, Cabrera M, Hernández P, Boiani L, Lavaggi ML, Di Maio R, Yaluff G, Serna E, Torres S, Ferreira ME, Vera de Bilbao N, Torres E, Pérez-Silanes S, Solano B, Moreno E, Aldana I, López de Ceráin A, Cerecetto H, González M, Monge A. Benitez D, et al. J Med Chem. 2011 May 26;54(10):3624-36. doi: 10.1021/jm2002469. Epub 2011 May 4. J Med Chem. 2011. PMID: 21506600
Helietta apiculata: a tropical weapon against Chagas disease.
Elena Ferreira M, Rojas de Arias A, Yaluff G, Vera de Bilbao N, Nakayama H, Torres S, Schinini A, Torres S, Serna E, Torrecilhas AC, Fournet A, Cebrián-Torrejón G. Elena Ferreira M, et al. Nat Prod Res. 2019 Nov;33(22):3308-3311. doi: 10.1080/14786419.2018.1472594. Epub 2018 May 10. Nat Prod Res. 2019. PMID: 29745731
Zanthoxylum chiloperone leaves extract: first sustainable Chagas disease treatment.
Ferreira ME, Cebrián-Torrejón G, Corrales AS, Vera de Bilbao N, Rolón M, Gomez CV, Leblanc K, Yaluf G, Schinini A, Torres S, Serna E, Rojas de Arias A, Poupon E, Fournet A. Ferreira ME, et al. J Ethnopharmacol. 2011 Feb 16;133(3):986-93. doi: 10.1016/j.jep.2010.11.032. Epub 2010 Dec 4. J Ethnopharmacol. 2011. PMID: 21134431
13 results