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Hybridization Approach Toward Novel Antituberculars: Design, Synthesis, and Biological Evaluation of Compounds Combining Pyrazinamide and 4-Aminosalicylic Acid.
Bouz G, Šlechta P, Jand'ourek O, Konečná K, Paterová P, Bárta P, Novák M, Kučera R, Dal NK, Fenaroli F, Zemanová J, Forbak M, Korduláková J, Pavliš O, Kubíčková P, Doležal M, Zitko J. Bouz G, et al. Among authors: pavlis o. ACS Infect Dis. 2023 Jan 13;9(1):79-96. doi: 10.1021/acsinfecdis.2c00433. Epub 2022 Dec 28. ACS Infect Dis. 2023. PMID: 36577009
Bispecific antibody neutralizes circulating SARS-CoV-2 variants, prevents escape and protects mice from disease.
De Gasparo R, Pedotti M, Simonelli L, Nickl P, Muecksch F, Cassaniti I, Percivalle E, Lorenzi JCC, Mazzola F, Magrì D, Michalcikova T, Haviernik J, Honig V, Mrazkova B, Polakova N, Fortova A, Tureckova J, Iatsiuk V, Girolamo SD, Palus M, Zudova D, Bednar P, Bukova I, Bianchini F, Mehn D, Nencka R, Strakova P, Pavlis O, Rozman J, Gioria S, Camilla Sammartino J, Giardina F, Gaiarsa S, Hammarström QP, Barnes CO, Bjorkman PJ, Calzolai L, Piralla A, Baldanti F, Nussenzweig MC, Bieniasz PD, Hatziioannou T, Prochazka J, Sedlacek R, Robbiani DF, Ruzek D, Varani L. De Gasparo R, et al. Among authors: pavlis o. bioRxiv [Preprint]. 2021 Mar 5:2021.01.22.427567. doi: 10.1101/2021.01.22.427567. bioRxiv. 2021. PMID: 33501434 Free PMC article. Preprint.
Our experience using real-time PCR for the detection of the gene that encodes the superficial lipoprotein LipL32 of the pathogenic leptospires to confirm the acute form of human leptospirosis.
Kucerova P, Cermakova Z, Pliskova L, Pavlis O, Kubickova P, Kleprlikova H, Valenta Z. Kucerova P, et al. Among authors: pavlis o. Biomed Pap Med Fac Univ Palacky Olomouc Czech Repub. 2013 Dec;157(4):387-91. doi: 10.5507/bp.2012.109. Epub 2012 Dec 7. Biomed Pap Med Fac Univ Palacky Olomouc Czech Repub. 2013. PMID: 23235722 Free article.
S-substituted 3,5-dinitrophenyl 1,3,4-oxadiazole-2-thiols and tetrazole-5-thiols as highly efficient antitubercular agents.
Karabanovich G, Němeček J, Valášková L, Carazo A, Konečná K, Stolaříková J, Hrabálek A, Pavliš O, Pávek P, Vávrová K, Roh J, Klimešová V. Karabanovich G, et al. Among authors: pavlis o. Eur J Med Chem. 2017 Jan 27;126:369-383. doi: 10.1016/j.ejmech.2016.11.041. Epub 2016 Nov 21. Eur J Med Chem. 2017. PMID: 27907875
Rifampicin Nanoformulation Enhances Treatment of Tuberculosis in Zebrafish.
Trousil J, Syrová Z, Dal NK, Rak D, Konefał R, Pavlova E, Matějková J, Cmarko D, Kubíčková P, Pavliš O, Urbánek T, Sedlák M, Fenaroli F, Raška I, Štěpánek P, Hrubý M. Trousil J, et al. Among authors: pavlis o. Biomacromolecules. 2019 Apr 8;20(4):1798-1815. doi: 10.1021/acs.biomac.9b00214. Epub 2019 Mar 6. Biomacromolecules. 2019. PMID: 30785284
Development of 3,5-Dinitrophenyl-Containing 1,2,4-Triazoles and Their Trifluoromethyl Analogues as Highly Efficient Antitubercular Agents Inhibiting Decaprenylphosphoryl-β-d-ribofuranose 2'-Oxidase.
Karabanovich G, Dušek J, Savková K, Pavliš O, Pávková I, Korábečný J, Kučera T, Kočová Vlčková H, Huszár S, Konyariková Z, Konečná K, Jand'ourek O, Stolaříková J, Korduláková J, Vávrová K, Pávek P, Klimešová V, Hrabálek A, Mikušová K, Roh J. Karabanovich G, et al. Among authors: pavlis o. J Med Chem. 2019 Sep 12;62(17):8115-8139. doi: 10.1021/acs.jmedchem.9b00912. Epub 2019 Aug 22. J Med Chem. 2019. PMID: 31393122
Antimycobacterial pyridine carboxamides: From design to in vivo activity.
Nawrot DE, Bouz G, Janďourek O, Konečná K, Paterová P, Bárta P, Novák M, Kučera R, Zemanová J, Forbak M, Korduláková J, Pavliš O, Kubíčková P, Doležal M, Zitko J. Nawrot DE, et al. Among authors: pavlis o. Eur J Med Chem. 2023 Oct 5;258:115617. doi: 10.1016/j.ejmech.2023.115617. Epub 2023 Jun 30. Eur J Med Chem. 2023. PMID: 37423128 Free article.
29 results