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Optimisation of pyrazolo[1,5-a]pyrimidin-7(4H)-one derivatives as novel Hsp90 C-terminal domain inhibitors against Ewing sarcoma.
Bioorg Chem. 2023 Feb;131:106311. doi: 10.1016/j.bioorg.2022.106311. Epub 2022 Dec 5.
Bioorg Chem. 2023.
PMID: 36495678
Free article.
Discovery of Novel Hsp90 C-Terminal Inhibitors Using 3D-Pharmacophores Derived from Molecular Dynamics Simulations.
Tomašič T, Durcik M, Keegan BM, Skledar DG, Zajec Ž, Blagg BSJ, Bryant SD.
Tomašič T, et al. Among authors: zajec z.
Int J Mol Sci. 2020 Sep 20;21(18):6898. doi: 10.3390/ijms21186898.
Int J Mol Sci. 2020.
PMID: 32962253
Free PMC article.
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Structure-Activity Relationships of Benzothiazole-Based Hsp90 C-Terminal-Domain Inhibitors.
Dernovšek J, Zajec Ž, Durcik M, Mašič LP, Gobec M, Zidar N, Tomašič T.
Dernovšek J, et al. Among authors: zajec z.
Pharmaceutics. 2021 Aug 17;13(8):1283. doi: 10.3390/pharmaceutics13081283.
Pharmaceutics. 2021.
PMID: 34452244
Free PMC article.
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In Silico Discovery and Optimisation of a Novel Structural Class of Hsp90 C-Terminal Domain Inhibitors.
Zajec Ž, Dernovšek J, Gobec M, Tomašič T.
Zajec Ž, et al.
Biomolecules. 2022 Jun 24;12(7):884. doi: 10.3390/biom12070884.
Biomolecules. 2022.
PMID: 35883440
Free PMC article.
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Catalytic Stereoconvergent Synthesis of Homochiral β-CF3, β-SCF3, and β-OCF3 Benzylic Alcohols.
Cotman AE, Dub PA, Sterle M, Lozinšek M, Dernovšek J, Zajec Ž, Zega A, Tomašič T, Cahard D.
Cotman AE, et al. Among authors: zajec z.
ACS Org Inorg Au. 2022 Oct 5;2(5):396-404. doi: 10.1021/acsorginorgau.2c00019. Epub 2022 Jun 8.
ACS Org Inorg Au. 2022.
PMID: 36217345
Free PMC article.
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ATP-competitive inhibitors of human DNA topoisomerase IIα with improved antiproliferative activity based on N-phenylpyrrolamide scaffold.
Skok Ž, Durcik M, Zajec Ž, Gramec Skledar D, Bozovičar K, Pišlar A, Tomašič T, Zega A, Peterlin Mašič L, Kikelj D, Zidar N, Ilaš J.
Skok Ž, et al. Among authors: zajec z.
Eur J Med Chem. 2023 Mar 5;249:115116. doi: 10.1016/j.ejmech.2023.115116. Epub 2023 Jan 18.
Eur J Med Chem. 2023.
PMID: 36689894
Free article.
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Refined high-content imaging-based phenotypic drug screening in zebrafish xenografts.
Sturtzel C, Grissenberger S, Bozatzi P, Scheuringer E, Wenninger-Weinzierl A, Zajec Z, Dernovšek J, Pascoal S, Gehl V, Kutsch A, Granig A, Rifatbegovic F, Carre M, Lang A, Valtingojer I, Moll J, Lötsch D, Erhart F, Widhalm G, Surdez D, Delattre O, André N, Stampfl J, Tomašič T, Taschner-Mandl S, Distel M.
Sturtzel C, et al. Among authors: zajec z.
NPJ Precis Oncol. 2023 May 18;7(1):44. doi: 10.1038/s41698-023-00386-9.
NPJ Precis Oncol. 2023.
PMID: 37202469
Free PMC article.
Review.
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Workplace noise exposure after modernisation of an aluminium processing complex.
Doko-Jelinić J, Lukić J, Udovicić R, Zuskin E, Nola IA, Zajec Z.
Doko-Jelinić J, et al. Among authors: zajec z.
Arh Hig Rada Toksikol. 2009 Sep;60(3):343-8. doi: 10.2478/10004-1254-60-2009-1902.
Arh Hig Rada Toksikol. 2009.
PMID: 19789164
Free article.
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