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A new D₂ dopamine receptor agonist allosterically modulates A(2A) adenosine receptor signalling by interacting with the A(2A)/D₂ receptor heteromer.
Trincavelli ML, Daniele S, Orlandini E, Navarro G, Casadó V, Giacomelli C, Nencetti S, Nuti E, Macchia M, Huebner H, Gmeiner P, Rossello A, Lluís C, Martini C. Trincavelli ML, et al. Cell Signal. 2012 Apr;24(4):951-60. doi: 10.1016/j.cellsig.2011.12.018. Epub 2011 Dec 30. Cell Signal. 2012. PMID: 22230688
Modulation of A2B adenosine receptor by 1-Benzyl-3-ketoindole derivatives.
Taliani S, Trincavelli ML, Cosimelli B, Laneri S, Severi E, Barresi E, Pugliesi I, Daniele S, Giacomelli C, Greco G, Novellino E, Martini C, Da Settimo F. Taliani S, et al. Among authors: trincavelli ml. Eur J Med Chem. 2013 Nov;69:331-7. doi: 10.1016/j.ejmech.2013.09.001. Epub 2013 Sep 8. Eur J Med Chem. 2013. PMID: 24077183
Apoptosis therapy in cancer: the first single-molecule co-activating p53 and the translocator protein in glioblastoma.
Daniele S, Taliani S, Da Pozzo E, Giacomelli C, Costa B, Trincavelli ML, Rossi L, La Pietra V, Barresi E, Carotenuto A, Limatola A, Lamberti A, Marinelli L, Novellino E, Da Settimo F, Martini C. Daniele S, et al. Among authors: trincavelli ml. Sci Rep. 2014 Apr 23;4:4749. doi: 10.1038/srep04749. Sci Rep. 2014. PMID: 24756113 Free PMC article.
Further studies on pyrazolo[1',5':1,6]pyrimido[4,5-d]pyridazin-4(3H)-ones as potent and selective human A1 adenosine receptor antagonists.
Giovannoni MP, Ciciani G, Cilibrizzi A, Crocetti L, Daniele S, Di Cesare Mannelli L, Ghelardini C, Giacomelli C, Guerrini G, Martini C, Trincavelli ML, Vergelli C. Giovannoni MP, et al. Among authors: trincavelli ml. Eur J Med Chem. 2015 Jan 7;89:32-41. doi: 10.1016/j.ejmech.2014.10.020. Epub 2014 Oct 12. Eur J Med Chem. 2015. PMID: 25462223
♦Copper (II) ions modulate Angiogenin activity in human endothelial cells.
Giacomelli C, Trincavelli ML, Satriano C, Hansson Ö, La Mendola D, Rizzarelli E, Martini C. Giacomelli C, et al. Among authors: trincavelli ml. Int J Biochem Cell Biol. 2015 Mar;60:185-96. doi: 10.1016/j.biocel.2015.01.005. Epub 2015 Jan 14. Int J Biochem Cell Biol. 2015. PMID: 25596488
Toward PET imaging of A2B adenosine receptors: a carbon-11 labeled triazinobenzimidazole tracer: Synthesis and imaging of a new A2B PET tracer.
Petroni D, Giacomelli C, Taliani S, Barresi E, Robello M, Daniele S, Bartoli A, Burchielli S, Pardini S, Salvadori PA, Da Settimo F, Martini C, Trincavelli ML, Menichetti L. Petroni D, et al. Among authors: trincavelli ml. Nucl Med Biol. 2016 May;43(5):309-17. doi: 10.1016/j.nucmedbio.2016.02.005. Epub 2016 Feb 27. Nucl Med Biol. 2016. PMID: 27150034
115 results