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Stereoselective synthesis of 3,4-dihydropyrrolo[1,2-a]pyrazin-1(2H)-one derivatives as PIM kinase inhibitors inspired from marine alkaloids.
Chirality. 2022 Nov;34(11):1437-1452. doi: 10.1002/chir.23501. Epub 2022 Aug 12.
Chirality. 2022.
PMID: 35959859
The generation of purinome-targeted libraries as a means to diversify ATP-mimetic chemical classes for lead finding.
Felder ER, Badari A, Disingrini T, Mantegani S, Orrenius C, Avanzi N, Isacchi A, Salom B.
Felder ER, et al. Among authors: disingrini t.
Mol Divers. 2012 Feb;16(1):27-51. doi: 10.1007/s11030-012-9361-6. Epub 2012 Feb 15.
Mol Divers. 2012.
PMID: 22350112
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Synthesis and SAR of new pyrazolo[4,3-h]quinazoline-3-carboxamide derivatives as potent and selective MPS1 kinase inhibitors.
Caldarelli M, Angiolini M, Disingrini T, Donati D, Guanci M, Nuvoloni S, Posteri H, Quartieri F, Silvagni M, Colombo R.
Caldarelli M, et al. Among authors: disingrini t.
Bioorg Med Chem Lett. 2011 Aug 1;21(15):4507-11. doi: 10.1016/j.bmcl.2011.05.122. Epub 2011 Jun 14.
Bioorg Med Chem Lett. 2011.
PMID: 21723120
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Design, synthesis, and action of oxotremorine-related hybrid-type allosteric modulators of muscarinic acetylcholine receptors.
Disingrini T, Muth M, Dallanoce C, Barocelli E, Bertoni S, Kellershohn K, Mohr K, De Amici M, Holzgrabe U.
Disingrini T, et al.
J Med Chem. 2006 Jan 12;49(1):366-72. doi: 10.1021/jm050769s.
J Med Chem. 2006.
PMID: 16392821
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Dualsteric GPCR targeting: a novel route to binding and signaling pathway selectivity.
Antony J, Kellershohn K, Mohr-Andrä M, Kebig A, Prilla S, Muth M, Heller E, Disingrini T, Dallanoce C, Bertoni S, Schrobang J, Tränkle C, Kostenis E, Christopoulos A, Höltje HD, Barocelli E, De Amici M, Holzgrabe U, Mohr K.
Antony J, et al. Among authors: disingrini t.
FASEB J. 2009 Feb;23(2):442-50. doi: 10.1096/fj.08-114751. Epub 2008 Oct 8.
FASEB J. 2009.
PMID: 18842964
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