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Stereoselective synthesis of 3,4-dihydropyrrolo[1,2-a]pyrazin-1(2H)-one derivatives as PIM kinase inhibitors inspired from marine alkaloids.
Chirality. 2022 Nov;34(11):1437-1452. doi: 10.1002/chir.23501. Epub 2022 Aug 12.
Chirality. 2022.
PMID: 35959859
Discovery and optimization of pyrrolo[1,2-a]pyrazinones leads to novel and selective inhibitors of PIM kinases.
Casuscelli F, Ardini E, Avanzi N, Casale E, Cervi G, D'Anello M, Donati D, Faiardi D, Ferguson RD, Fogliatto G, Galvani A, Marsiglio A, Mirizzi DG, Montemartini M, Orrenius C, Papeo G, Piutti C, Salom B, Felder ER.
Casuscelli F, et al.
Bioorg Med Chem. 2013 Dec 1;21(23):7364-80. doi: 10.1016/j.bmc.2013.09.054. Epub 2013 Oct 2.
Bioorg Med Chem. 2013.
PMID: 24139169
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Fragment-based hit discovery and structure-based optimization of aminotriazoloquinazolines as novel Hsp90 inhibitors.
Casale E, Amboldi N, Brasca MG, Caronni D, Colombo N, Dalvit C, Felder ER, Fogliatto G, Galvani A, Isacchi A, Polucci P, Riceputi L, Sola F, Visco C, Zuccotto F, Casuscelli F.
Casale E, et al. Among authors: casuscelli f.
Bioorg Med Chem. 2014 Aug 1;22(15):4135-50. doi: 10.1016/j.bmc.2014.05.056. Epub 2014 Jun 14.
Bioorg Med Chem. 2014.
PMID: 24980703
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Structure-based optimization of potent PDK1 inhibitors.
Angiolini M, Banfi P, Casale E, Casuscelli F, Fiorelli C, Saccardo MB, Silvagni M, Zuccotto F.
Angiolini M, et al. Among authors: casuscelli f.
Bioorg Med Chem Lett. 2010 Jul 15;20(14):4095-9. doi: 10.1016/j.bmcl.2010.05.070. Epub 2010 Jun 8.
Bioorg Med Chem Lett. 2010.
PMID: 20621725
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The Novel PIM1 Inhibitor NMS-P645 Reverses PIM1-Dependent Effects on TMPRSS2/ERG Positive Prostate Cancer Cells And Shows Anti-Proliferative Activity in Combination with PI3K Inhibition.
Mologni L, Magistroni V, Casuscelli F, Montemartini M, Gambacorti-Passerini C.
Mologni L, et al. Among authors: casuscelli f.
J Cancer. 2017 Jan 1;8(1):140-145. doi: 10.7150/jca.15838. eCollection 2017.
J Cancer. 2017.
PMID: 28123608
Free PMC article.
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Study of the compositional changes of mango during ripening by use of nuclear magnetic resonance spectroscopy.
Gil AM, Duarte IF, Delgadillo I, Colquhoun IJ, Casuscelli F, Humpfer E, Spraul M.
Gil AM, et al. Among authors: casuscelli f.
J Agric Food Chem. 2000 May;48(5):1524-36. doi: 10.1021/jf9911287.
J Agric Food Chem. 2000.
PMID: 10820054
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Isolation and characterization of Guiera senegalensis J.F.Gmel. active principles.
Ficarra R, Ficarra P, Tommasini S, Carulli M, Melardi S, Di Bella MR, Calabrò ML, De Pasquale R, Germanò MP, Sanogo R, Casuscelli F.
Ficarra R, et al. Among authors: casuscelli f.
Boll Chim Farm. 1997 May;136(5):454-9.
Boll Chim Farm. 1997.
PMID: 9281895
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Genetically epilepsy-prone rodents show some changes of ion levels in the brain.
Saija A, Princi P, Casuscelli F, Lanza M, Scalese M, Trombetta D, Costa G, De Sarro G.
Saija A, et al. Among authors: casuscelli f.
Brain Res Bull. 1994;33(1):1-6. doi: 10.1016/0361-9230(94)90043-4.
Brain Res Bull. 1994.
PMID: 8275321
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