Szymańska E - Search Results

1

Discovery of the First Highly Selective Antagonist of the GluK3 Kainate Receptor Subtype.

Chałupnik P, Vialko A, Pickering DS, Hinkkanen M, Donbosco S, Møller TC, Jensen AA, Nielsen B, Bay Y, Kristensen AS, Johansen TN, Łątka K, Bajda M, Szymańska E. Chałupnik P, et al. Among authors: szymanska e. Int J Mol Sci. 2022 Aug 8;23(15):8797. doi: 10.3390/ijms23158797. Int J Mol Sci. 2022. PMID: 35955932 Free PMC article.

2

3-Substituted phenylalanines as selective AMPA- and kainate receptor ligands.

Szymańska E, Pickering DS, Nielsen B, Johansen TN. Szymańska E, et al. Bioorg Med Chem. 2009 Sep 1;17(17):6390-401. doi: 10.1016/j.bmc.2009.07.021. Epub 2009 Jul 16. Bioorg Med Chem. 2009. PMID: 19656686

3

A new phenylalanine derivative acts as an antagonist at the AMPA receptor GluA2 and introduces partial domain closure: synthesis, resolution, pharmacology, and crystal structure.

Szymańska E, Frydenvang K, Contreras-Sanz A, Pickering DS, Frola E, Serafimoska Z, Nielsen B, Kastrup JS, Johansen TN. Szymańska E, et al. J Med Chem. 2011 Oct 27;54(20):7289-98. doi: 10.1021/jm200862h. Epub 2011 Oct 4. J Med Chem. 2011. PMID: 21923187

4

Structural and pharmacological characterization of phenylalanine-based AMPA receptor antagonists at kainate receptors.

Venskutonytė R, Frydenvang K, Valadés EA, Szymańska E, Johansen TN, Kastrup JS, Pickering DS. Venskutonytė R, et al. Among authors: szymanska e. ChemMedChem. 2012 Oct;7(10):1793-8. doi: 10.1002/cmdc.201100599. Epub 2012 Mar 7. ChemMedChem. 2012. PMID: 22407805

5

Discovery of novel lead in the group of N-substituted piperazine ether derivatives with potential histamine H3 receptor activity.

Kuder KJ, Stachnik M, Schunack W, Szymańska E, Kieć-Kononowicz K. Kuder KJ, et al. Among authors: szymanska e. Med Chem. 2014;10(6):588-99. doi: 10.2174/15734064113096660050. Med Chem. 2014. PMID: 24047214

6

Studies on Aryl-Substituted Phenylalanines: Synthesis, Activity, and Different Binding Modes at AMPA Receptors.

Szymanska E, Frydenvang K, Pickering DS, Krintel C, Nielsen B, Kooshki A, Zachariassen LG, Olsen L, Kastrup JS, Johansen TN. Szymanska E, et al. J Med Chem. 2016 Jan 14;59(1):448-61. doi: 10.1021/acs.jmedchem.5b01666. Epub 2015 Dec 22. J Med Chem. 2016. PMID: 26653877

7

Design, synthesis and structure-activity relationships of novel phenylalanine-based amino acids as kainate receptors ligands.

Szymańska E, Chałupnik P, Szczepańska K, Cuñado Moral AM, Pickering DS, Nielsen B, Johansen TN, Kieć-Kononowicz K. Szymańska E, et al. Bioorg Med Chem Lett. 2016 Nov 15;26(22):5568-5572. doi: 10.1016/j.bmcl.2016.09.075. Epub 2016 Sep 30. Bioorg Med Chem Lett. 2016. PMID: 27765511

8

Aryl- and heteroaryl-substituted phenylalanines as AMPA receptor ligands.

Szymańska E, Chałupnik P, Johansen TN, Nielsen B, Cuñado Moral AM, Pickering DS, Więckowska A, Kieć-Kononowicz K. Szymańska E, et al. Chem Biol Drug Des. 2017 Dec;90(6):1271-1281. doi: 10.1111/cbdd.13048. Epub 2017 Jul 18. Chem Biol Drug Des. 2017. PMID: 28636281

9

Pharmacological characterization and binding modes of novel racemic and optically active phenylalanine-based antagonists of AMPA receptors.

Szymańska E, Nielsen B, Johansen TN, Cuñado Moral AM, Pickering DS, Szczepańska K, Mickowska A, Kieć-Kononowicz K. Szymańska E, et al. Eur J Med Chem. 2017 Sep 29;138:874-883. doi: 10.1016/j.ejmech.2017.07.007. Epub 2017 Jul 8. Eur J Med Chem. 2017. PMID: 28738307

10

5-Arylidenerhodanines as P-gp Modulators: An Interesting Effect of the Carboxyl Group on ABCB1 Function in Multidrug-Resistant Cancer Cells.

Żesławska E, Tejchman W, Kincses A, Spengler G, Nitek W, Żuchowski G, Szymańska E. Żesławska E, et al. Among authors: szymanska e. Int J Mol Sci. 2022 Sep 16;23(18):10812. doi: 10.3390/ijms231810812. Int J Mol Sci. 2022. PMID: 36142724 Free PMC article.

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