Kristensen AS - Search Results

1

Discovery of the First Highly Selective Antagonist of the GluK3 Kainate Receptor Subtype.

Chałupnik P, Vialko A, Pickering DS, Hinkkanen M, Donbosco S, Møller TC, Jensen AA, Nielsen B, Bay Y, Kristensen AS, Johansen TN, Łątka K, Bajda M, Szymańska E. Chałupnik P, et al. Among authors: kristensen as. Int J Mol Sci. 2022 Aug 8;23(15):8797. doi: 10.3390/ijms23158797. Int J Mol Sci. 2022. PMID: 35955932 Free PMC article.

2

Design, synthesis, and pharmacology of a highly subtype-selective GluR1/2 agonist, (RS)-2-amino-3-(4-chloro-3-hydroxy-5-isoxazolyl)propionic acid (Cl-HIBO).

Bjerrum EJ, Kristensen AS, Pickering DS, Greenwood JR, Nielsen B, Liljefors T, Schousboe A, Bräuner-Osborne H, Madsen U. Bjerrum EJ, et al. Among authors: kristensen as. J Med Chem. 2003 May 22;46(11):2246-9. doi: 10.1021/jm020588f. J Med Chem. 2003. PMID: 12747796

3

Synthesis and in vitro pharmacology at AMPA and kainate preferring glutamate receptors of 4-heteroarylmethylidene glutamate analogues.

Valgeirsson J, Christensen JK, Kristensen AS, Pickering DS, Nielsen B, Fischer CH, Bräuner-Osborne H, Nielsen EØ, Krogsgaard-Larsen P, Madsen U. Valgeirsson J, et al. Among authors: kristensen as. Bioorg Med Chem. 2003 Oct 1;11(20):4341-9. doi: 10.1016/s0968-0896(03)00485-1. Bioorg Med Chem. 2003. PMID: 13129570

4

2-arylureidobenzoic acids: selective noncompetitive antagonists for the homomeric kainate receptor subtype GluR5.

Valgeirsson J, Nielsen EØ, Peters D, Varming T, Mathiesen C, Kristensen AS, Madsen U. Valgeirsson J, et al. Among authors: kristensen as. J Med Chem. 2003 Dec 18;46(26):5834-43. doi: 10.1021/jm030428j. J Med Chem. 2003. PMID: 14667236

5

The structure of a mixed GluR2 ligand-binding core dimer in complex with (S)-glutamate and the antagonist (S)-NS1209.

Kasper C, Pickering DS, Mirza O, Olsen L, Kristensen AS, Greenwood JR, Liljefors T, Schousboe A, Wätjen F, Gajhede M, Sigurskjold BW, Kastrup JS. Kasper C, et al. Among authors: kristensen as. J Mol Biol. 2006 Apr 7;357(4):1184-201. doi: 10.1016/j.jmb.2006.01.024. Epub 2006 Jan 31. J Mol Biol. 2006. PMID: 16483599

6

Ionotropic glutamate-like receptor delta2 binds D-serine and glycine.

Naur P, Hansen KB, Kristensen AS, Dravid SM, Pickering DS, Olsen L, Vestergaard B, Egebjerg J, Gajhede M, Traynelis SF, Kastrup JS. Naur P, et al. Among authors: kristensen as. Proc Natl Acad Sci U S A. 2007 Aug 28;104(35):14116-21. doi: 10.1073/pnas.0703718104. Epub 2007 Aug 21. Proc Natl Acad Sci U S A. 2007. PMID: 17715062 Free PMC article.

7

The glutamate receptor GluR5 agonist (S)-2-amino-3-(3-hydroxy-7,8-dihydro-6H-cyclohepta[d]isoxazol-4-yl)propionic acid and the 8-methyl analogue: synthesis, molecular pharmacology, and biostructural characterization.

Clausen RP, Naur P, Kristensen AS, Greenwood JR, Strange M, Bräuner-Osborne H, Jensen AA, Nielsen AS, Geneser U, Ringgaard LM, Nielsen B, Pickering DS, Brehm L, Gajhede M, Krogsgaard-Larsen P, Kastrup JS. Clausen RP, et al. Among authors: kristensen as. J Med Chem. 2009 Aug 13;52(15):4911-22. doi: 10.1021/jm900565c. J Med Chem. 2009. PMID: 19588945

8

Evaluation of PhTX-74 as subtype-selective inhibitor of GluA2-containing AMPA receptors.

Poulsen MH, Lucas S, Strømgaard K, Kristensen AS. Poulsen MH, et al. Among authors: kristensen as. Mol Pharmacol. 2014 Feb;85(2):261-8. doi: 10.1124/mol.113.089961. Epub 2013 Nov 12. Mol Pharmacol. 2014. PMID: 24220009

9

Analogues of 3-hydroxyisoxazole-containing glutamate receptor ligands based on the 3-hydroxypyrazole-moiety: design, synthesis and pharmacological characterization.

Jørgensen L, Nielsen B, Pickering DS, Kristensen AS, Frydenvang K, Madsen U, Clausen RP. Jørgensen L, et al. Among authors: kristensen as. Neurochem Res. 2014 Oct;39(10):1895-905. doi: 10.1007/s11064-014-1332-0. Epub 2014 May 22. Neurochem Res. 2014. PMID: 24848194

10

Pharmacology and Structural Analysis of Ligand Binding to the Orthosteric Site of Glutamate-Like GluD2 Receptors.

Kristensen AS, Hansen KB, Naur P, Olsen L, Kurtkaya NL, Dravid SM, Kvist T, Yi F, Pøhlsgaard J, Clausen RP, Gajhede M, Kastrup JS, Traynelis SF. Kristensen AS, et al. Mol Pharmacol. 2016 Feb;89(2):253-62. doi: 10.1124/mol.115.100909. Epub 2015 Dec 10. Mol Pharmacol. 2016. PMID: 26661043 Free PMC article.

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