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Functionalized Allopurinols Targeting Amyloid-Binding Alcohol Dehydrogenase Rescue Aβ-Induced Mitochondrial Dysfunction.
ACS Chem Neurosci. 2022 Jul 20;13(14):2176-2190. doi: 10.1021/acschemneuro.2c00246. Epub 2022 Jul 8.
ACS Chem Neurosci. 2022.
PMID: 35802826
The evolution of small molecule enzyme activators.
Dow LF, Case AM, Paustian MP, Pinkerton BR, Simeon P, Trippier PC.
Dow LF, et al.
RSC Med Chem. 2023 Sep 22;14(11):2206-2230. doi: 10.1039/d3md00399j. eCollection 2023 Nov 15.
RSC Med Chem. 2023.
PMID: 37974956
Review.
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Discovery of an Aldo-Keto reductase 1C3 (AKR1C3) degrader.
Carmona AV, Jonnalagadda S, Case AM, Maddeboina K, Jonnalagadda SK, Dow LF, Duan L, Penning TM, Trippier PC.
Carmona AV, et al. Among authors: dow lf.
Commun Chem. 2024 Apr 29;7(1):95. doi: 10.1038/s42004-024-01177-4.
Commun Chem. 2024.
PMID: 38684887
Free PMC article.
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