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The NLRP3 Inflammasome Pathway: A Review of Mechanisms and Inhibitors for the Treatment of Inflammatory Diseases.
Front Aging Neurosci. 2022 Jun 10;14:879021. doi: 10.3389/fnagi.2022.879021. eCollection 2022.
Front Aging Neurosci. 2022.
PMID: 35754962
Free PMC article.
Review.
Development of bivalent compounds as potential neuroprotectants for Alzheimer's disease.
He L, Jiang Y, Green J, Blevins H, Zhang S.
He L, et al.
Bioorg Med Chem Lett. 2019 Aug 1;29(15):1957-1961. doi: 10.1016/j.bmcl.2019.05.035. Epub 2019 May 18.
Bioorg Med Chem Lett. 2019.
PMID: 31153803
Free PMC article.
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Discovery of Second-Generation NLRP3 Inflammasome Inhibitors: Design, Synthesis, and Biological Characterization.
Jiang Y, He L, Green J, Blevins H, Guo C, Patel SH, Halquist MS, McRae M, Venitz J, Wang XY, Zhang S.
Jiang Y, et al.
J Med Chem. 2019 Nov 14;62(21):9718-9731. doi: 10.1021/acs.jmedchem.9b01155. Epub 2019 Oct 31.
J Med Chem. 2019.
PMID: 31626545
Free PMC article.
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Discovery of carbon-11 labeled sulfonamide derivative: A PET tracer for imaging brain NLRP3 inflammasome.
Xu Y, Xu Y, Blevins H, Lan Y, Liu Y, Yuan G, Striar R, Zagaroli JS, Tocci DR, Langan AG, Zhang C, Zhang S, Wang C.
Xu Y, et al.
Bioorg Med Chem Lett. 2021 Feb 15;34:127777. doi: 10.1016/j.bmcl.2021.127777. Epub 2021 Jan 6.
Bioorg Med Chem Lett. 2021.
PMID: 33418063
Free PMC article.
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A Novel Inhibitor Targeting NLRP3 Inflammasome Reduces Neuropathology and Improves Cognitive Function in Alzheimer's Disease Transgenic Mice.
Kuwar R, Rolfe A, Di L, Blevins H, Xu Y, Sun X, Bloom GS, Zhang S, Sun D.
Kuwar R, et al.
J Alzheimers Dis. 2021;82(4):1769-1783. doi: 10.3233/JAD-210400.
J Alzheimers Dis. 2021.
PMID: 34219728
Free PMC article.
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Development of sulfonamide-based NLRP3 inhibitors: Further modifications and optimization through structure-activity relationship studies.
Xu Y, Xu Y, Blevins H, Guo C, Biby S, Wang XY, Wang C, Zhang S.
Xu Y, et al.
Eur J Med Chem. 2022 Aug 5;238:114468. doi: 10.1016/j.ejmech.2022.114468. Epub 2022 May 21.
Eur J Med Chem. 2022.
PMID: 35635948
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CPT1A-mediated fatty acid oxidation confers cancer cell resistance to immune-mediated cytolytic killing.
Liu Z, Liu W, Wang W, Ma Y, Wang Y, Drum DL, Cai J, Blevins H, Lee E, Shah S, Fisher PB, Wang X, Fang X, Guo C, Wang XY.
Liu Z, et al.
Proc Natl Acad Sci U S A. 2023 Sep 26;120(39):e2302878120. doi: 10.1073/pnas.2302878120. Epub 2023 Sep 18.
Proc Natl Acad Sci U S A. 2023.
PMID: 37722058
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