Discovery of a potent and selective proteolysis targeting chimera (PROTAC) degrader of NSD3 histone methyltransferase.
Sun Y, Zhang Y, Chen X, Yu A, Du W, Huang Y, Wu F, Yu L, Li J, Wen C, Yang H, Shi Q, Geng M, Huang X, Xu S.
Sun Y, et al. Among authors: li j.
Eur J Med Chem. 2022 Sep 5;239:114528. doi: 10.1016/j.ejmech.2022.114528. Epub 2022 Jun 13.
Eur J Med Chem. 2022.
PMID: 35717870