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Exploring Aspartic Protease Inhibitor Binding to Design Selective Antimalarials.
J Chem Inf Model. 2022 Jul 11;62(13):3263-3273. doi: 10.1021/acs.jcim.2c00422. Epub 2022 Jun 17.
J Chem Inf Model. 2022.
PMID: 35712895
A Polymorphism in leuS Confers Reduced Susceptibility to GSK2251052 in a Clinical Isolate of Staphylococcus aureus.
Gupta A, Monteferrante C, Rasina D, Leitis G, Randall CP, Tomlinson JH, Jirgensons A, Goessens WH, Hays JP, O'Neill AJ.
Gupta A, et al. Among authors: leitis g.
Antimicrob Agents Chemother. 2016 Apr 22;60(5):3219-21. doi: 10.1128/AAC.02940-15. Print 2016 May.
Antimicrob Agents Chemother. 2016.
PMID: 26976861
Free PMC article.
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Azole-based non-peptidomimetic plasmepsin inhibitors.
Kinena L, Leitis G, Kanepe-Lapsa I, Bobrovs R, Jaudzems K, Ozola V, Suna E, Jirgensons A.
Kinena L, et al. Among authors: leitis g.
Arch Pharm (Weinheim). 2018 Sep;351(9):e1800151. doi: 10.1002/ardp.201800151. Epub 2018 Jul 31.
Arch Pharm (Weinheim). 2018.
PMID: 30063266
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Synthesis and evaluation of an agrocin 84 toxic moiety (TM84) analogue as a malarial threonyl tRNA synthetase inhibitor.
Buitrago JAR, Leitis G, Kaņepe-Lapsa I, Rudnickiha A, Parisini E, Jirgensons A.
Buitrago JAR, et al. Among authors: leitis g.
Org Biomol Chem. 2023 Jul 5;21(26):5433-5439. doi: 10.1039/d3ob00670k.
Org Biomol Chem. 2023.
PMID: 37335076
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Spiropyran-Based Photoisomerizable α-Amino Acid for Membrane-Active Peptide Modification.
Hrebonkin A, Afonin S, Nikitjuka A, Borysov OV, Leitis G, Babii O, Koniev S, Lorig T, Grage SL, Nick P, Ulrich AS, Jirgensons A, Komarov IV.
Hrebonkin A, et al. Among authors: leitis g.
Chemistry. 2024 Apr 16;30(22):e202400066. doi: 10.1002/chem.202400066. Epub 2024 Mar 1.
Chemistry. 2024.
PMID: 38366887
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