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Discovery of novel SARS-CoV-2 inhibitors targeting the main protease Mpro by virtual screenings and hit optimization.
Antiviral Res. 2022 Aug;204:105350. doi: 10.1016/j.antiviral.2022.105350. Epub 2022 Jun 7.
Antiviral Res. 2022.
PMID: 35688349
Free PMC article.
Indomethacin-based PROTACs as pan-coronavirus antiviral agents.
Desantis J, Mercorelli B, Celegato M, Croci F, Bazzacco A, Baroni M, Siragusa L, Cruciani G, Loregian A, Goracci L.
Desantis J, et al. Among authors: bazzacco a.
Eur J Med Chem. 2021 Dec 15;226:113814. doi: 10.1016/j.ejmech.2021.113814. Epub 2021 Sep 4.
Eur J Med Chem. 2021.
PMID: 34534839
Free PMC article.
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Design, synthesis, and biological evaluation of first-in-class indomethacin-based PROTACs degrading SARS-CoV-2 main protease and with broad-spectrum antiviral activity.
Desantis J, Bazzacco A, Eleuteri M, Tuci S, Bianconi E, Macchiarulo A, Mercorelli B, Loregian A, Goracci L.
Desantis J, et al. Among authors: bazzacco a.
Eur J Med Chem. 2024 Mar 15;268:116202. doi: 10.1016/j.ejmech.2024.116202. Epub 2024 Feb 6.
Eur J Med Chem. 2024.
PMID: 38394929
Free article.
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On the production of ancient Egyptian blue: Multi-modal characterization and micron-scale luminescence mapping.
Seymour LM, Nicola M, Kessler MI, Yost CL, Bazzacco A, Marello A, Ferraris E, Gobetto R, Masic A.
Seymour LM, et al. Among authors: bazzacco a.
PLoS One. 2020 Nov 24;15(11):e0242549. doi: 10.1371/journal.pone.0242549. eCollection 2020.
PLoS One. 2020.
PMID: 33232351
Free PMC article.
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