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Structure‒tissue exposure/selectivity relationship (STR) correlates with clinical efficacy/safety.
Acta Pharm Sin B. 2022 May;12(5):2462-2478. doi: 10.1016/j.apsb.2022.02.015. Epub 2022 Feb 23.
Acta Pharm Sin B. 2022.
PMID: 35646532
Free PMC article.
A gastrointestinal locally activating Janus kinase inhibitor to treat ulcerative colitis.
Bu Y, Traore MDM, Zhang L, Wang L, Liu Z, Hu H, Wang M, Li C, Sun D.
Bu Y, et al. Among authors: traore mdm.
J Biol Chem. 2023 Dec;299(12):105467. doi: 10.1016/j.jbc.2023.105467. Epub 2023 Nov 17.
J Biol Chem. 2023.
PMID: 37979913
Free PMC article.
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Crossing of the Cystic Barriers of Toxoplasma gondii by the Fluorescent Coumarin Tetra-Cyclopeptide.
Dard C, Leforestier B, Francisco Hilário F, Traoré MDM, Lespinasse MA, Pérès B, Molina MC, Pereira de Freitas R, Milet A, Maubon D, Wong YS.
Dard C, et al. Among authors: traore mdm.
Molecules. 2021 Dec 11;26(24):7506. doi: 10.3390/molecules26247506.
Molecules. 2021.
PMID: 34946588
Free PMC article.
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Hydroxyl Ketone-Based Histone Deacetylase Inhibitors To Gain Insight into Class I HDAC Selectivity versus That of HDAC6.
Traoré MDM, Zwick V, Simões-Pires CA, Nurisso A, Issa M, Cuendet M, Maynadier M, Wein S, Vial H, Jamet H, Wong YS.
Traoré MDM, et al.
ACS Omega. 2017 Apr 30;2(4):1550-1562. doi: 10.1021/acsomega.6b00481. Epub 2017 Apr 20.
ACS Omega. 2017.
PMID: 30023639
Free PMC article.
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Synthesis of an Uncharged Tetra-cyclopeptide Acting as a Transmembrane Carrier: Enhanced Cellular and Nuclear Uptake.
Francisco Hilário F, Traoré MD, Zwick V, Berry L, Simões-Pires CA, Cuendet M, Fantozzi N, Pereira de Freitas R, Maynadier M, Wein S, Vial H, Wong YS.
Francisco Hilário F, et al.
Org Lett. 2017 Feb 3;19(3):612-615. doi: 10.1021/acs.orglett.6b03776. Epub 2017 Jan 20.
Org Lett. 2017.
PMID: 28107021
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