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From cycloheptathiophene-3-carboxamide to oxazinone-based derivatives as allosteric HIV-1 ribonuclease H inhibitors.
Massari S, Corona A, Distinto S, Desantis J, Caredda A, Sabatini S, Manfroni G, Felicetti T, Cecchetti V, Pannecouque C, Maccioni E, Tramontano E, Tabarrini O. Massari S, et al. Among authors: desantis j. J Enzyme Inhib Med Chem. 2019 Dec;34(1):55-74. doi: 10.1080/14756366.2018.1523901. J Enzyme Inhib Med Chem. 2019. PMID: 30362381 Free PMC article.
Antitubercular polyhalogenated phenothiazines and phenoselenazine with reduced binding to CNS receptors.
Nizi MG, Desantis J, Nakatani Y, Massari S, Mazzarella MA, Shetye G, Sabatini S, Barreca ML, Manfroni G, Felicetti T, Rushton-Green R, Hards K, Latacz G, Satała G, Bojarski AJ, Cecchetti V, Kolář MH, Handzlik J, Cook GM, Franzblau SG, Tabarrini O. Nizi MG, et al. Among authors: desantis j. Eur J Med Chem. 2020 Sep 1;201:112420. doi: 10.1016/j.ejmech.2020.112420. Epub 2020 Jun 5. Eur J Med Chem. 2020. PMID: 32526553
A Broad Anti-influenza Hybrid Small Molecule That Potently Disrupts the Interaction of Polymerase Acidic Protein-Basic Protein 1 (PA-PB1) Subunits.
Massari S, Nannetti G, Desantis J, Muratore G, Sabatini S, Manfroni G, Mercorelli B, Cecchetti V, Palù G, Cruciani G, Loregian A, Goracci L, Tabarrini O. Massari S, et al. Among authors: desantis j. J Med Chem. 2015 May 14;58(9):3830-42. doi: 10.1021/acs.jmedchem.5b00012. Epub 2015 Apr 20. J Med Chem. 2015. PMID: 25856229 Free article.
Indomethacin-based PROTACs as pan-coronavirus antiviral agents.
Desantis J, Mercorelli B, Celegato M, Croci F, Bazzacco A, Baroni M, Siragusa L, Cruciani G, Loregian A, Goracci L. Desantis J, et al. Eur J Med Chem. 2021 Dec 15;226:113814. doi: 10.1016/j.ejmech.2021.113814. Epub 2021 Sep 4. Eur J Med Chem. 2021. PMID: 34534839 Free PMC article.
Proteolysis targeting chimeras in antiviral research.
Desantis J, Goracci L. Desantis J, et al. Future Med Chem. 2022 Apr;14(7):459-462. doi: 10.4155/fmc-2022-0005. Epub 2022 Feb 8. Future Med Chem. 2022. PMID: 35134309 No abstract available.
76 results