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Potentiation of antibiotic activity, and efflux pumps inhibition by (2E)-1-(4-aminophenyl)-3-(4-fluorophenyl)prop-2-en-1-one.
Fundam Clin Pharmacol. 2022 Dec;36(6):1066-1082. doi: 10.1111/fcp.12785. Epub 2022 May 19.
Fundam Clin Pharmacol. 2022.
PMID: 35475507
Antibacterial and antibiotic modifying activity of chalcone (2E)-1-(4'-aminophenyl)-3-(4-methoxyphenyl)-prop-2-en-1-one in strains of Staphylococcus aureus carrying NorA and MepA efflux pumps: In vitro and in silico approaches.
Silva J, Esmeraldo Rocha J, da Cunha Xavier J, Sampaio de Freitas T, Douglas Melo Coutinho H, Nogueira Bandeira P, Rodrigues de Oliveira M, Nunes da Rocha M, Machado Marinho E, de Kassio Vieira Monteiro N, Ribeiro LR, Róseo Paula Pessoa Bezerra de Menezes R, Machado Marinho M, Magno Rodrigues Teixeira A, Silva Dos Santos H, Silva Marinho E.
Silva J, et al. Among authors: magno rodrigues teixeira a.
Microb Pathog. 2022 Aug;169:105664. doi: 10.1016/j.micpath.2022.105664. Epub 2022 Jul 5.
Microb Pathog. 2022.
PMID: 35803497
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In silico study of the potential interactions of 4'-acetamidechalcones with protein targets in SARS-CoV-2.
Q Almeida-Neto FW, Castro Matos MG, Marinho EM, Marinho MM, Róseo Paula Pessoa Bezerra de Menezes R, Sampaio TL, Bandeira PN, Celedonio Fernandes CF, Magno Rodrigues Teixeira A, Marinho ES, de Lima-Neto P, Silva Dos Santos H.
Q Almeida-Neto FW, et al. Among authors: magno rodrigues teixeira a.
Biochem Biophys Res Commun. 2021 Jan 22;537:71-77. doi: 10.1016/j.bbrc.2020.12.074. Epub 2020 Dec 26.
Biochem Biophys Res Commun. 2021.
PMID: 33387885
Free PMC article.
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