Nefzi A - Search Results

1

1,5-Disubstituted Acylated 2-Amino-4,5-dihydroimidazoles as a New Class of Retinoic Acid Receptor-Related Orphan Receptor (ROR) Inhibitors.

Ortiz MA, Piedrafita FJ, Nefzi A. Ortiz MA, et al. Among authors: nefzi a. Int J Mol Sci. 2022 Apr 17;23(8):4433. doi: 10.3390/ijms23084433. Int J Mol Sci. 2022. PMID: 35457251 Free PMC article.

2

Diversity oriented synthesis and IKK inhibition of aminobenzimidazole tethered quinazoline-2,4-diones, thioxoquinazolin-4-ones, benzodiazepine-2,3,5-triones, isoxazoles and isoxazolines.

Dadiboyena S, Arfaoui A, Amri H, Piedrafita FJ, Nefzi A. Dadiboyena S, et al. Among authors: nefzi a. Bioorg Med Chem Lett. 2015 Feb 1;25(3):685-9. doi: 10.1016/j.bmcl.2014.11.078. Epub 2014 Dec 8. Bioorg Med Chem Lett. 2015. PMID: 25522820 Free PMC article.

3

Synthesis of dihydroimidazole tethered imidazolinethiones and their activity as novel antagonists of the nuclear retinoic acid receptor-related orphan receptors (RORs).

Nefzi A, Marconi GD, Ortiz MA, Davis JC, Piedrafita FJ. Nefzi A, et al. Bioorg Med Chem Lett. 2017 Apr 1;27(7):1608-1610. doi: 10.1016/j.bmcl.2017.02.014. Epub 2017 Feb 10. Bioorg Med Chem Lett. 2017. PMID: 28242276 Free PMC article.

4

Discovery of cyclic guanidine-linked sulfonamides as inhibitors of LMTK3 kinase.

Ortiz MA, Michaels H, Molina B, Toenjes S, Davis J, Marconi GD, Hecht D, Gustafson JL, Piedrafita FJ, Nefzi A. Ortiz MA, et al. Among authors: nefzi a. Bioorg Med Chem Lett. 2020 May 1;30(9):127108. doi: 10.1016/j.bmcl.2020.127108. Epub 2020 Mar 17. Bioorg Med Chem Lett. 2020. PMID: 32192797

5

Small Molecule Compounds Identified from Mixture-Based Library Inhibit Binding between Plasmodium falciparum Infected Erythrocytes and Endothelial Receptor ICAM-1.

Chesnokov O, Visitdesotrakul P, Kalani K, Nefzi A, Oleinikov AV. Chesnokov O, et al. Among authors: nefzi a. Int J Mol Sci. 2021 May 26;22(11):5659. doi: 10.3390/ijms22115659. Int J Mol Sci. 2021. PMID: 34073419 Free PMC article.

6

Bis-Cyclic Guanidine Heterocyclic Peptidomimetics as Opioid Ligands with Mixed μ-, κ- and δ-Opioid Receptor Interactions: A Potential Approach to Novel Analgesics.

McLaughlin JP, Rayala R, Bunnell AJ, Tantak MP, Eans SO, Nefzi K, Ganno ML, Dooley CT, Nefzi A. McLaughlin JP, et al. Among authors: nefzi a. Int J Mol Sci. 2022 Aug 25;23(17):9623. doi: 10.3390/ijms23179623. Int J Mol Sci. 2022. PMID: 36077029 Free PMC article.

7

Integrating computational and mixture-based screening of combinatorial libraries.

Yongye AB, Pinilla C, Medina-Franco JL, Giulianotti MA, Dooley CT, Appel JR, Nefzi A, Scior T, Houghten RA, Martínez-Mayorga K. Yongye AB, et al. Among authors: nefzi a. J Mol Model. 2011 Jun;17(6):1473-82. doi: 10.1007/s00894-010-0850-1. Epub 2010 Sep 21. J Mol Model. 2011. PMID: 20853183

8

Potent antimicrobial small molecules screened as inhibitors of tyrosine recombinases and Holliday junction-resolving enzymes.

Rideout MC, Boldt JL, Vahi-Ferguson G, Salamon P, Nefzi A, Ostresh JM, Giulianotti M, Pinilla C, Segall AM. Rideout MC, et al. Among authors: nefzi a. Mol Divers. 2011 Nov;15(4):989-1005. doi: 10.1007/s11030-011-9333-2. Epub 2011 Sep 22. Mol Divers. 2011. PMID: 21938393

9

Scaffold ranking and positional scanning utilized in the discovery of nAChR-selective compounds suitable for optimization studies.

Wu J, Zhang Y, Maida LE, Santos RG, Welmaker GS, LaVoi TM, Nefzi A, Yu Y, Houghten RA, Toll L, Giulianotti MA. Wu J, et al. Among authors: nefzi a. J Med Chem. 2013 Dec 27;56(24):10103-17. doi: 10.1021/jm401543h. Epub 2013 Dec 12. J Med Chem. 2013. PMID: 24274400 Free PMC article.

10

Integrating virtual screening and combinatorial chemistry for accelerated drug discovery.

López-Vallejo F, Caulfield T, Martínez-Mayorga K, Giulianotti MA, Nefzi A, Houghten RA, Medina-Franco JL. López-Vallejo F, et al. Among authors: nefzi a. Comb Chem High Throughput Screen. 2011 Jul;14(6):475-87. doi: 10.2174/138620711795767866. Comb Chem High Throughput Screen. 2011. PMID: 21521151 Review.

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