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Overcoming Paradoxical Kinase Priming by a Novel MNK1 Inhibitor.
J Med Chem. 2022 Apr 28;65(8):6070-6087. doi: 10.1021/acs.jmedchem.1c01941. Epub 2022 Apr 13.
J Med Chem. 2022.
PMID: 35417652
Free PMC article.
C4-C5 fused pyrazol-3-amines: when the degree of unsaturation and electronic characteristics of the fused ring controls regioselectivity in Ullmann and acylation reactions.
Bou-Petit E, Plans A, Rodríguez-Picazo N, Torres-Coll A, Puigjaner C, Font-Bardia M, Teixidó J, Ramon Y Cajal S, Estrada-Tejedor R, Borrell JI.
Bou-Petit E, et al.
Org Biomol Chem. 2020 Jul 15;18(27):5145-5156. doi: 10.1039/d0ob00796j.
Org Biomol Chem. 2020.
PMID: 32583833
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Mutated RAS-associating proteins and ERK activation in relapse/refractory diffuse large B cell lymphoma.
Benoit A, Bou-Petit E, Chou H, Lu M, Guilbert C, Luo VM, Assouline S, Morin RD, Dmitrienko S, Estrada-Tejedor R, Johnson NA, Mann KK.
Benoit A, et al. Among authors: bou petit e.
Sci Rep. 2022 Jan 17;12(1):779. doi: 10.1038/s41598-021-04736-0.
Sci Rep. 2022.
PMID: 35039569
Free PMC article.
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