Discovery of a highly potent CECR2 bromodomain inhibitor with 7H-pyrrolo[2,3-d] pyrimidine scaffold.
Lu H, Lu T, Zu S, Duan Z, Guang Y, Li Q, Ma J, Chen D, Li B, Lu W, Jiang H, Luo C, Ye D, Chen K, Lin H.
Lu H, et al. Among authors: chen k, chen d.
Bioorg Chem. 2022 Jun;123:105768. doi: 10.1016/j.bioorg.2022.105768. Epub 2022 Mar 26.
Bioorg Chem. 2022.
PMID: 35378372