Rutjes FPJT - Search Results

1

Cyclobutanes in Small-Molecule Drug Candidates.

van der Kolk MR, Janssen MACH, Rutjes FPJT, Blanco-Ania D. van der Kolk MR, et al. ChemMedChem. 2022 May 4;17(9):e202200020. doi: 10.1002/cmdc.202200020. Epub 2022 Mar 29. ChemMedChem. 2022. PMID: 35263505 Free PMC article. Review.

2

Solution-phase parallel annulation of (thio)hydantoins to tetrahydroisoquinolines and tetrahydro-beta-carbolines containing the 2-arylethyl amine scaffold.

Blanco-Ania D, Hermkens PH, Sliedregt LA, Scheeren HW, Rutjes FP. Blanco-Ania D, et al. J Comb Chem. 2009 Jul-Aug;11(4):547-55. doi: 10.1021/cc8001926. J Comb Chem. 2009. PMID: 19472984

3

Synthesis of hydantoins and thiohydantoins spiro-fused to pyrrolidines: druglike molecules based on the 2-arylethyl amine scaffold.

Blanco-Ania D, Hermkens PH, Sliedregt LA, Scheeren HW, Rutjes FP. Blanco-Ania D, et al. J Comb Chem. 2009 Jul-Aug;11(4):527-38. doi: 10.1021/cc800190z. J Comb Chem. 2009. PMID: 19472985

4

Synthesis of tetrahydro-beta-carbolines and tetrahydroisoquinolines fused to pyrrolidines and solution-phase parallel acylation.

Blanco-Ania D, Hermkens PH, Sliedregt LA, Scheeren HW, Rutjes FP. Blanco-Ania D, et al. J Comb Chem. 2009 Jul-Aug;11(4):539-46. doi: 10.1021/cc800191w. J Comb Chem. 2009. PMID: 19472986

5

Synthesis of dihydrouracils spiro-fused to pyrrolidines: druglike molecules based on the 2-arylethyl amine scaffold.

Blanco-Ania D, Valderas-Cortina C, Hermkens PH, Sliedregt LA, Scheeren HW, Rutjes FP. Blanco-Ania D, et al. Molecules. 2010 Mar 30;15(4):2269-301. doi: 10.3390/molecules15042269. Molecules. 2010. PMID: 20428042 Free PMC article.

6

Oxidation of Secondary Methyl Ethers to Ketones.

Gilissen PJ, Blanco-Ania D, Rutjes FPJT. Gilissen PJ, et al. J Org Chem. 2017 Jul 7;82(13):6671-6679. doi: 10.1021/acs.joc.7b00632. Epub 2017 Jun 12. J Org Chem. 2017. PMID: 28585818 Free PMC article.

7

Pd-Catalyzed Hydroamination of Alkoxyallenes with Azole Heterocycles: Examples and Mechanistic Proposal.

Bernar I, Fiser B, Blanco-Ania D, Gómez-Bengoa E, Rutjes FPJT. Bernar I, et al. Org Lett. 2017 Aug 18;19(16):4211-4214. doi: 10.1021/acs.orglett.7b01826. Epub 2017 Aug 8. Org Lett. 2017. PMID: 28786679 Free PMC article.

8

Trifluoromethyl Vinyl Sulfide: A Building Block for the Synthesis of CF₃S-Containing Isoxazolidines.

Riesco-Domínguez A, van de Wiel J, Hamlin TA, van Beek B, Lindell SD, Blanco-Ania D, Bickelhaupt FM, Rutjes FPJT. Riesco-Domínguez A, et al. J Org Chem. 2018 Feb 16;83(4):1779-1789. doi: 10.1021/acs.joc.7b02639. Epub 2018 Jan 30. J Org Chem. 2018. PMID: 29320179 Free PMC article.

9

Structure-Activity Relationship Studies on (R)-PFI-2 Analogues as Inhibitors of Histone Lysine Methyltransferase SETD7.

Lenstra DC, Damen E, Leenders RGG, Blaauw RH, Rutjes FPJT, Wegert A, Mecinović J. Lenstra DC, et al. ChemMedChem. 2018 Jul 18;13(14):1405-1413. doi: 10.1002/cmdc.201800242. Epub 2018 Jun 25. ChemMedChem. 2018. PMID: 29869845

10

Carbonylonium ions: the onium ions of the carbonyl group.

Blanco-Ania D, Rutjes FPJT. Blanco-Ania D, et al. Beilstein J Org Chem. 2018 Oct 4;14:2568-2571. doi: 10.3762/bjoc.14.233. eCollection 2018. Beilstein J Org Chem. 2018. PMID: 30410617 Free PMC article.

Save citations to file

Email citations

Send citations to clipboard

Add to Collections

Add to My Bibliography

Create a file for external citation management software

Your saved search

Your RSS Feed

My NCBI Filters

Text availability

Article attribute

Article type

Publication date

188 results

Search Page