Björkling F - Search Results

1

Synthesis and Structure-Activity Relationships of Novel Non-Steroidal CYP17A1 Inhibitors as Potential Prostate Cancer Agents.

Wróbel TM, Rogova O, Sharma K, Rojas Velazquez MN, Pandey AV, Jørgensen FS, Arendrup FS, Andersen KL, Björkling F. Wróbel TM, et al. Among authors: bjorkling f. Biomolecules. 2022 Jan 20;12(2):165. doi: 10.3390/biom12020165. Biomolecules. 2022. PMID: 35204665 Free PMC article.

2

Nicotinamide phosphoribosyltransferase inhibitors, design, preparation, and structure-activity relationship.

Christensen MK, Erichsen KD, Olesen UH, Tjørnelund J, Fristrup P, Thougaard A, Nielsen SJ, Sehested M, Jensen PB, Loza E, Kalvinsh I, Garten A, Kiess W, Björkling F. Christensen MK, et al. Among authors: bjorkling f. J Med Chem. 2013 Nov 27;56(22):9071-88. doi: 10.1021/jm4009949. Epub 2013 Nov 13. J Med Chem. 2013. PMID: 24164086

3

Discovery of Novel Non-Steroidal Cytochrome P450 17A1 Inhibitors as Potential Prostate Cancer Agents.

Wróbel TM, Rogova O, Andersen KL, Yadav R, Brixius-Anderko S, Scott EE, Olsen L, Jørgensen FS, Björkling F. Wróbel TM, et al. Among authors: bjorkling f. Int J Mol Sci. 2020 Jul 9;21(14):4868. doi: 10.3390/ijms21144868. Int J Mol Sci. 2020. PMID: 32660148 Free PMC article.

4

Non-steroidal CYP17A1 Inhibitors: Discovery and Assessment.

Wróbel TM, Jørgensen FS, Pandey AV, Grudzińska A, Sharma K, Yakubu J, Björkling F. Wróbel TM, et al. Among authors: bjorkling f. J Med Chem. 2023 May 25;66(10):6542-6566. doi: 10.1021/acs.jmedchem.3c00442. Epub 2023 May 16. J Med Chem. 2023. PMID: 37191389 Free PMC article. Review.

5

Exploring the Potential of Sulfur Moieties in Compounds Inhibiting Steroidogenesis.

Wróbel TM, Sharma K, Mannella I, Oliaro-Bosso S, Nieckarz P, Du Toit T, Voegel CD, Rojas Velazquez MN, Yakubu J, Matveeva A, Therkelsen S, Jørgensen FS, Pandey AV, Pippione AC, Lolli ML, Boschi D, Björkling F. Wróbel TM, et al. Among authors: bjorkling f. Biomolecules. 2023 Sep 5;13(9):1349. doi: 10.3390/biom13091349. Biomolecules. 2023. PMID: 37759751 Free PMC article.

6

Synthesis and structure-activity relationship of aminobenzophenones. A novel class of p38 MAP kinase inhibitors with high antiinflammatory activity.

Ottosen ER, Sørensen MD, Björkling F, Skak-Nielsen T, Fjording MS, Aaes H, Binderup L. Ottosen ER, et al. Among authors: bjorkling f. J Med Chem. 2003 Dec 18;46(26):5651-62. doi: 10.1021/jm030851s. J Med Chem. 2003. PMID: 14667219

7

Synthesis and antitumor effect in vitro and in vivo of substituted 1,3-dihydroindole-2-ones.

Christensen MK, Erichsen KD, Trojel-Hansen C, Tjørnelund J, Nielsen SJ, Frydenvang K, Johansen TN, Nielsen B, Sehested M, Jensen PB, Ikaunieks M, Zaichenko A, Loza E, Kalvinsh I, Björkling F. Christensen MK, et al. Among authors: bjorkling f. J Med Chem. 2010 Oct 14;53(19):7140-5. doi: 10.1021/jm100763j. J Med Chem. 2010. PMID: 20845961

8

Novel Agonist Bioisosteres and Common Structure-Activity Relationships for The Orphan G Protein-Coupled Receptor GPR139.

Shehata MA, Nøhr AC, Lissa D, Bisig C, Isberg V, Andersen KB, Harpsøe K, Björkling F, Bräuner-Osborne H, Gloriam DE. Shehata MA, et al. Among authors: bjorkling f. Sci Rep. 2016 Nov 10;6:36681. doi: 10.1038/srep36681. Sci Rep. 2016. PMID: 27830715 Free PMC article.

9

Binding of alpha-hydroxy-beta-amino acid inhibitors to methionine aminopeptidase. The performance of two types of scoring functions.

Jørgensen AT, Sørensen MD, Björkling F, Liljefors T. Jørgensen AT, et al. Among authors: bjorkling f. J Comput Aided Mol Des. 2003 May-Jun;17(5-6):383-97. doi: 10.1023/a:1026149810619. J Comput Aided Mol Des. 2003. PMID: 14635729

10

Novel amide derivatives as inhibitors of histone deacetylase: design, synthesis and SAR.

Andrianov V, Gailite V, Lola D, Loza E, Semenikhina V, Kalvinsh I, Finn P, Petersen KD, Ritchie JW, Khan N, Tumber A, Collins LS, Vadlamudi SM, Björkling F, Sehested M. Andrianov V, et al. Among authors: bjorkling f. Eur J Med Chem. 2009 Mar;44(3):1067-85. doi: 10.1016/j.ejmech.2008.06.020. Epub 2008 Jun 27. Eur J Med Chem. 2009. PMID: 18672316

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