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Illuminating a Dark Kinase: Structure-Guided Design, Synthesis, and Evaluation of a Potent Nek1 Inhibitor and Its Effects on the Embryonic Zebrafish Pronephros.
J Med Chem. 2022 Jan 27;65(2):1265-1282. doi: 10.1021/acs.jmedchem.0c02118. Epub 2021 Mar 16.
J Med Chem. 2022.
PMID: 35081715
Design, synthesis and biological evaluation of novel aminopyrazole- and 7-azaindole-based Nek1 inhibitors and their effects on zebrafish kidney development.
Pilakowski J, Baumann G, Shih YH, Meckel T, Schmidt B.
Pilakowski J, et al.
Bioorg Med Chem Lett. 2021 Dec 1;53:128418. doi: 10.1016/j.bmcl.2021.128418. Epub 2021 Oct 26.
Bioorg Med Chem Lett. 2021.
PMID: 34715306
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Structure-based optimization of oxadiazole-based GSK-3 inhibitors.
Lo Monte F, Kramer T, Gu J, Brodrecht M, Pilakowski J, Fuertes A, Dominguez JM, Plotkin B, Eldar-Finkelman H, Schmidt B.
Lo Monte F, et al. Among authors: pilakowski j.
Eur J Med Chem. 2013 Mar;61:26-40. doi: 10.1016/j.ejmech.2012.06.006. Epub 2012 Jun 12.
Eur J Med Chem. 2013.
PMID: 22749643
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