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Page 1
Synthesis, in vitro and in vivo pharmacological evaluation of serotoninergic ligands containing an isonicotinic nucleus.
Fiorino F, Ciano A, Magli E, Severino B, Corvino A, Perissutti E, Frecentese F, Di Vaio P, Izzo AA, Capasso R, Massarelli P, Nencini C, Rossi I, Kędzierska E, Orzelska-Gòrka J, Bielenica A, Santagada V, Caliendo G. Fiorino F, et al. Among authors: corvino a. Eur J Med Chem. 2016 Mar 3;110:133-50. doi: 10.1016/j.ejmech.2016.01.021. Epub 2016 Jan 18. Eur J Med Chem. 2016. PMID: 26820556
5-HT2 receptor affinity, docking studies and pharmacological evaluation of a series of 1,3-disubstituted thiourea derivatives.
Bielenica A, Kędzierska E, Koliński M, Kmiecik S, Koliński A, Fiorino F, Severino B, Magli E, Corvino A, Rossi I, Massarelli P, Kozioł AE, Sawczenko A, Struga M. Bielenica A, et al. Among authors: corvino a. Eur J Med Chem. 2016 Jun 30;116:173-186. doi: 10.1016/j.ejmech.2016.03.073. Epub 2016 Mar 30. Eur J Med Chem. 2016. PMID: 27061981
Synthesis of Arylpiperazine Derivatives as Protease Activated Receptor 1 Antagonists and Their Evaluation as Antiproliferative Agents.
Zotti AI, Di Gennaro E, Corvino A, Frecentese F, Magli E, Perissutti E, Cirino G, Roviezzo F, Terranova-Barberio M, Iannelli F, Caliendo G, Santagada V, Fiorino F, Budillon A, Severino B. Zotti AI, et al. Among authors: corvino a. Anticancer Agents Med Chem. 2017;17(7):973-981. doi: 10.2174/1871520616666160926120904. Anticancer Agents Med Chem. 2017. PMID: 27671294
Activity of human kallikrein-related peptidase 6 (KLK6) on substrates containing sequences of basic amino acids. Is it a processing protease?
Silva RN, Oliveira LCG, Parise CB, Oliveira JR, Severino B, Corvino A, di Vaio P, Temussi PA, Caliendo G, Santagada V, Juliano L, Juliano MA. Silva RN, et al. Among authors: corvino a. Biochim Biophys Acta Proteins Proteom. 2017 May;1865(5):558-564. doi: 10.1016/j.bbapap.2017.02.017. Epub 2017 Feb 28. Biochim Biophys Acta Proteins Proteom. 2017. PMID: 28254587
New 5-HT1A, 5HT2A and 5HT2C receptor ligands containing a picolinic nucleus: Synthesis, in vitro and in vivo pharmacological evaluation.
Fiorino F, Magli E, Kędzierska E, Ciano A, Corvino A, Severino B, Perissutti E, Frecentese F, Di Vaio P, Saccone I, Izzo AA, Capasso R, Massarelli P, Rossi I, Orzelska-Gòrka J, Kotlińska JH, Santagada V, Caliendo G. Fiorino F, et al. Among authors: corvino a. Bioorg Med Chem. 2017 Oct 15;25(20):5820-5837. doi: 10.1016/j.bmc.2017.09.018. Epub 2017 Sep 18. Bioorg Med Chem. 2017. PMID: 28943244
1,2,4-Thiadiazolidin-3,5-diones as novel hydrogen sulfide donors.
Severino B, Corvino A, Fiorino F, Luciano P, Frecentese F, Magli E, Saccone I, Di Vaio P, Citi V, Calderone V, Servillo L, Casale R, Cirino G, Vellecco V, Bucci M, Perissutti E, Santagada V, Caliendo G. Severino B, et al. Among authors: corvino a. Eur J Med Chem. 2018 Jan 1;143:1677-1686. doi: 10.1016/j.ejmech.2017.10.068. Epub 2017 Nov 11. Eur J Med Chem. 2018. PMID: 29133036
157 results