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Design, synthesis, structural optimization, SAR, in silico prediction of physicochemical properties and pharmacological evaluation of novel & potent thiazolo[4,5-d]pyrimidine corticotropin releasing factor (CRF) receptor antagonists.
Islam MR, Teleb M, Karageorgos V, Sakellaris S, Papadopoulos M, Pirmettis I, Fronczek FR, Liapakis G, Fahmy H. Islam MR, et al. Among authors: liapakis g. Eur J Pharm Sci. 2022 Feb 1;169:106084. doi: 10.1016/j.ejps.2021.106084. Epub 2021 Nov 29. Eur J Pharm Sci. 2022. PMID: 34856350 Free article.
Corticotrophin-Releasing Factor (CRF) and the urocortins are potent regulators of the inflammatory phenotype of human and mouse white adipocytes and the differentiation of mouse 3T3L1 pre-adipocytes.
Dermitzaki E, Liapakis G, Androulidaki A, Venihaki M, Melissas J, Tsatsanis C, Margioris AN. Dermitzaki E, et al. Among authors: liapakis g. PLoS One. 2014 May 16;9(5):e97060. doi: 10.1371/journal.pone.0097060. eCollection 2014. PLoS One. 2014. PMID: 24835211 Free PMC article.
Structural-functional analysis of the third transmembrane domain of the corticotropin-releasing factor type 1 receptor: role in activation and allosteric antagonism.
Spyridaki K, Matsoukas MT, Cordomi A, Gkountelias K, Papadokostaki M, Mavromoustakos T, Logothetis DE, Margioris AN, Pardo L, Liapakis G. Spyridaki K, et al. Among authors: liapakis g. J Biol Chem. 2014 Jul 4;289(27):18966-77. doi: 10.1074/jbc.M113.544460. Epub 2014 May 16. J Biol Chem. 2014. PMID: 24838244 Free PMC article.
69 results