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C6-structural optimizations of 2-aryl-1H-pyrazole-S-DABOs: From anti-HIV to anti-DENV activity.
Bioorg Chem. 2022 Feb;119:105494. doi: 10.1016/j.bioorg.2021.105494. Epub 2021 Nov 19.
Bioorg Chem. 2022.
PMID: 34836643
Synthesis and biological evaluation of a series of 2-(((5-akly/aryl-1H-pyrazol-3-yl)methyl)thio)-5-alkyl-6-(cyclohexylmethyl)-pyrimidin-4(3H)-ones as potential HIV-1 inhibitors.
Wu Y, Tang C, Rui R, Yang L, Ding W, Wang J, Li Y, Lai CC, Wang Y, Luo R, Xiao W, Zhang H, Zheng Y, He Y.
Wu Y, et al.
Acta Pharm Sin B. 2020 Mar;10(3):512-528. doi: 10.1016/j.apsb.2019.08.009. Epub 2019 Sep 5.
Acta Pharm Sin B. 2020.
PMID: 32140396
Free PMC article.
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